SCHEMBL2024918

SCHEMBL2024918

C[C@H]([C@H](O)c1ccccc1)N(C)C(=O)[C@@H](CC1CCOCC1)C(NC(=O)O)C(C)(C)C

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.41
NPY5R Q15761 12/20 0.38
NPY2R P49146 1/20 0.36
ALDH1A1 P00352 3/20 0.36
LMNA P02545 1/20 0.36
KDM4E B2RXH2 1/20 0.34
BRD4 O60885 1/20 0.34
HPGD P15428 1/20 0.34
TP53 P04637 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
NFKB1 P19838 1/20 0.34
MAPK1 P28482 1/20 0.34
CYP2C19 P33261 1/20 0.34
HIF1A Q16665 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8078131 0.77 GAA (0.43) GAANPY5RNPY2RALDH1A1KDM4E
SCHEMBL2024921 0.77 GAA (0.41) GAANPY5RNPY2RALDH1A1KDM4E
SCHEMBL2024919 0.77 GAA (0.41) GAANPY5RNPY2RALDH1A1KDM4E
SCHEMBL2028293 0.73 CNR1 (0.37)
SCHEMBL1107460 0.72 GAA (0.40) GAANPY5RNPY2RALDH1A1KDM4E
SCHEMBL8152205 0.70 GAA (0.51) GAANPY5RNPY2RALDH1A1KDM4E
SCHEMBL2668154 0.69 GAA (0.36) GAANPY5RNPY2RCYP3A4CYP2D6
SCHEMBL4380601 0.68 SLC6A4 (0.47) ALDH1A1LMNAKDM4EHPGDCYP3A4
SCHEMBL2020668 0.68 GAA (0.58) GAANPY5RNPY2RALDH1A1KDM4E
SCHEMBL7910584 0.67 PSEN1 (0.47) GAANPY5RALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110160300-A1 Renin Inhibitors and Methods of Use Thereof VITAE PHARMACEUTICALS, INC. 2011-06-30 US disclosed
US-20100160424-A1 RENIN INHIBITORS VITAE PHARMACEUTICALS, INC. 2010-06-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100160424-A1 RENIN INHIBITORS ACE, REN, DNPEP GAA 36/4885NPY5R 2086/4885NPY2R 2577/4885
US-20110160300-A1 Renin Inhibitors and Methods of Use Thereof REN, ACE, AGTR1 GAA 157/4885NPY5R 624/4885NPY2R 754/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.