SCHEMBL20249236

SCHEMBL20249236

CC(C)(C)c1ccc(N2CCCNCC2)cn1

nearest known ligand 0.62

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 16/20 0.62
CHRNA4 P43681 16/20 0.62
HTR1A P08908 1/20 0.48
HTR1D P28221 1/20 0.48
HTR1B P28222 1/20 0.48
HTR2A P28223 1/20 0.48
HTR7 P34969 1/20 0.48
HTR2B P41595 1/20 0.48
HTR3A P46098 1/20 0.48
HTR6 P50406 1/20 0.48
ADRB1 P08588 1/20 0.47
CHRNA1 P02708 1/20 0.44
CHRNA7 P36544 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12145921 0.94 CHRNB2 (0.58) CHRNB2CHRNA4HTR1AHTR1DHTR1B
SCHEMBL22601459 0.86 MAPT (0.50) CHRNB2CHRNA4
SCHEMBL16256660 0.84 MAPT (0.53) CHRNB2CHRNA4
SCHEMBL8108975 0.82 CHRNB2 (0.55) CHRNB2CHRNA4HTR3AHTR6ADRB1
Hydrochloric Acid SCHEMBL29978671 0.81 CHRNB2 (0.54) CHRNB2CHRNA4HTR3AHTR6ADRB1
Hydrochloric Acid SCHEMBL28343784 0.81 CHRNB2 (0.54) CHRNB2CHRNA4HTR3AHTR6ADRB1
SCHEMBL231910 0.80 CHRNB2 (0.68) CHRNB2CHRNA4ADRB1
SCHEMBL382350 0.78 CHRNB2 (0.58) CHRNB2CHRNA4HTR1DHTR3AHTR6
SCHEMBL31774414 0.78 CHRNB2 (0.58) CHRNB2CHRNA4HTR1DHTR3AHTR6
SCHEMBL20249102 0.77 CDK4 (0.43) CHRNB2CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180161329-A1 PYRIDO[3,4-D]PYRIMIDINE DERIVATIVE AND PHARMACEUTICALLY ACCEPTABLE SALT THEREOF TEIJIN PHARMA LIMITED (JP) 2018-06-14 US disclosed
US-20180161329-A1 PYRIDO[3,4-D]PYRIMIDINE DERIVATIVE AND PHARMACEUTICALLY ACCEPTABLE SALT THEREOF TEIJIN PHARMA LIMITED (JP) 2018-06-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180161329-A1 PYRIDO[3,4-D]PYRIMIDINE DERIVATIVE AND PHARMACEUTICALLY ACCEPTABLE SALT THEREOF CDK4, CDK6, CDK16 CHRNB2 4863/4885CHRNA4 4628/4885HTR1A 3202/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.