SCHEMBL8108975

SCHEMBL8108975

CC(C)(N)c1ccc(N2CCNCC2)cn1

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 9/20 0.55
CHRNA4 P43681 9/20 0.55
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47
LMNA P02545 1/20 0.47
ADRB1 P08588 4/20 0.46
AOC3 Q16853 1/20 0.43
HTR3E A5X5Y0 2/20 0.42
HTR3B O95264 2/20 0.42
HTR3A P46098 2/20 0.42
HTR3D Q70Z44 2/20 0.42
HTR3C Q8WXA8 2/20 0.42
SIGMAR1 Q99720 2/20 0.42
ADRB2 P07550 1/20 0.42
NCF1 P14598 1/20 0.42
PLD1 Q13393 1/20 0.42
HTR6 P50406 1/20 0.42
CDK4 P11802 1/20 0.41
CCND1 P24385 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12145921 0.87 CHRNB2 (0.58) CHRNB2CHRNA4KDM4EALDH1A1LMNA
Hydrochloric Acid SCHEMBL29978671 0.83 CHRNB2 (0.54) CHRNB2CHRNA4KDM4EALDH1A1LMNA
Hydrochloric Acid SCHEMBL28343784 0.83 CHRNB2 (0.54) CHRNB2CHRNA4KDM4EALDH1A1LMNA
SCHEMBL20249236 0.82 CHRNB2 (0.62) CHRNB2CHRNA4ADRB1HTR3AHTR6
SCHEMBL31774414 0.81 CHRNB2 (0.58) CHRNB2CHRNA4KDM4EALDH1A1LMNA
SCHEMBL382350 0.81 CHRNB2 (0.58) CHRNB2CHRNA4KDM4EALDH1A1LMNA
Hydrochloric Acid SCHEMBL382186 0.79 CHRNB2 (0.57) CHRNB2CHRNA4KDM4EALDH1A1LMNA
SCHEMBL1992377 0.75 CHRNB2 (0.64) CHRNB2CHRNA4KDM4EALDH1A1LMNA
SCHEMBL3917325 0.75 CHRNB2 (0.64) CHRNB2CHRNA4ADRB1HTR3EHTR3B
SCHEMBL20255149 0.74 CHRNB2 (0.44) CHRNB2CHRNA4CDK4CCND1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009001127-A1 CYANOCYCLOPROPYLCARBOXAMIDES AS CATHEPSIN INHIBITORS ASTRAZENECA AB (SE) 2008-12-31 WO disclosed