SCHEMBL20249390

SCHEMBL20249390

CC(C#N)N1CCN(c2ccc(C(C)(C)C)nc2)C(=O)C1

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 2/20 0.33
LGMN Q99538 1/20 0.32
HRH3 Q9Y5N1 2/20 0.31
TP53 P04637 1/20 0.31
DPP4 P27487 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20249308 0.87 HRH3 (0.38) IDH1HRH3TP53DPP4
SCHEMBL20255275 0.84 DRD3 (0.41) HRH3
SCHEMBL20249310 0.84 HRH3 (0.33) IDH1HRH3DPP4
SCHEMBL20249368 0.81 HRH3 (0.37) IDH1HRH3
SCHEMBL20249339 0.78 HRH3 (0.43) HRH3TP53
SCHEMBL20249366 0.78 ALDH1A1 (0.36) HRH3TP53DPP4
SCHEMBL20249115 0.77 SLC6A2 (0.42) HRH3TP53
SCHEMBL20249300 0.76 PIK3CD (0.43) IDH1HRH3DPP4
SCHEMBL20249342 0.74 PARP1 (0.35) HRH3
SCHEMBL20249159 0.74 DRD3 (0.33) TP53DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180161329-A1 PYRIDO[3,4-D]PYRIMIDINE DERIVATIVE AND PHARMACEUTICALLY ACCEPTABLE SALT THEREOF TEIJIN PHARMA LIMITED (JP) 2018-06-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180161329-A1 PYRIDO[3,4-D]PYRIMIDINE DERIVATIVE AND PHARMACEUTICALLY ACCEPTABLE SALT THEREOF CDK4, CDK6, CDK16 IDH1 147/4885LGMN 4798/4885HRH3 2304/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.