SCHEMBL20255201

SCHEMBL20255201

CC1(NC(=O)c2cc(Br)cnc2Cl)CC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ANO1 Q5XXA6 2/20 0.37
SORT1 Q99523 2/20 0.36
NPC1 O15118 2/20 0.36
MAPK1 P28482 2/20 0.36
RAB9A P51151 2/20 0.36
MAPT P10636 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
OPRK1 P41145 4/20 0.34
CNR2 P34972 2/20 0.34
FAAH O00519 1/20 0.34
HDAC3 O15379 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC2 Q92769 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
KDR P35968 3/20 0.34
TP53 P04637 1/20 0.33
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20241151 0.81 LRRK2 (0.42) ANO1NPC1RAB9AIRAK4
SCHEMBL30166593 0.81 LRRK2 (0.42) ANO1NPC1RAB9AIRAK4
SCHEMBL20254998 0.80 ANO1 (0.35) ANO1KDRPDE4APDE4BPDE4C
SCHEMBL15999441 0.80 OPRK1 (0.46) SORT1MAPTSMN1; SMN2OPRK1CNR2
SCHEMBL13555770 0.76 KDM4E (0.50) ANO1NPC1MAPK1RAB9ATP53
SCHEMBL13555773 0.75 BACE1 (0.42) HDAC3HDAC1HDAC2HDAC6
SCHEMBL20995140 0.75 BMPR1B (0.52) OPRK1CNR2
SCHEMBL20995143 0.75 BMPR1B (0.52) OPRK1CNR2
SCHEMBL30854837 0.75 CNR2 (0.51) NPC1RAB9ASMN1; SMN2OPRK1CNR2
SCHEMBL20240901 0.75 CNR2 (0.51) NPC1RAB9ASMN1; SMN2OPRK1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018104214-A1 METHOD FOR PRODUCING 5-(1-PHENYL-1H-PYRAZOLE-4-YL)-NICOTINAMIDE DERIVATIVES AND SIMILAR COMPOUNDS WITHOUT ISOLATING OR PURIFYING THE PHENYLHYDRAZINE INTERMEDIATE BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2018-06-14 WO disclosed