SCHEMBL20258331

SCHEMBL20258331

CC1=CC[C@@H]2CN(C)C[C@@H]2CC1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.40
SIGMAR1 Q99720 3/20 0.33
CHRNA7 P36544 2/20 0.30
MEN1 O00255 1/20 0.30
CYP3A4 P08684 1/20 0.30
ALOX15 P16050 1/20 0.30
MAPK1 P28482 1/20 0.30
KMT2A Q03164 1/20 0.30
STAT3 P40763 1/20 0.30
CHRNB2 P17787 1/20 0.30
CHRNB4 P30926 1/20 0.30
CHRNA3 P32297 1/20 0.30
CHRNA4 P43681 1/20 0.30
HRH3 Q9Y5N1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22305046 1.00 LMNA (0.40) LMNASIGMAR1CHRNA7MEN1CYP3A4
SCHEMBL20384069 0.79 TSHR (0.35)
SCHEMBL19788223 0.76 LMNA (0.33) LMNA
SCHEMBL20384101 0.73 SIGMAR1 (0.35) SIGMAR1MEN1CYP3A4ALOX15KMT2A
SCHEMBL20261092 0.69 LMNA (0.41) LMNACHRNA7MEN1CYP3A4ALOX15
SCHEMBL23508979 0.69 SIGMAR1 (0.35) SIGMAR1MEN1CYP3A4ALOX15KMT2A
SCHEMBL11444225 0.68 LMNA (0.40) LMNACHRNA7MEN1CYP3A4ALOX15
SCHEMBL12891347 0.68 LMNA (0.40) LMNACHRNA7MEN1CYP3A4ALOX15
SCHEMBL27397885 0.68 HRH3 (0.30) HRH3
SCHEMBL14627262 0.67 SIGMAR1 (0.46) SIGMAR1MEN1CYP3A4ALOX15KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018107112-A1 QUINOLONE-BASED COMPOUNDS WITH ANTICANCER ACTIVITY UNIVERSITY OF IOWA RESEARCH FOUNDATION (US) 2018-06-14 WO disclosed