SCHEMBL2026285

SCHEMBL2026285

Cc1cc(C(N)=O)ccc1-c1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.55
MKNK1 Q9BUB5 4/20 0.48
CHEK2 O96017 2/20 0.48
MKNK2 Q9HBH9 3/20 0.47
HSD17B1 P14061 1/20 0.47
PARP1 P09874 2/20 0.47
BCAT2 O15382 1/20 0.47
L3MBTL1 Q9Y468 2/20 0.47
POLB P06746 1/20 0.47
CYP3A4 P08684 1/20 0.47
MAPT P10636 1/20 0.47
TSHR P16473 1/20 0.47
CYP2C19 P33261 1/20 0.47
RECQL P46063 1/20 0.47
BLM P54132 1/20 0.47
PMP22 Q01453 1/20 0.47
HSD17B10 Q99714 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
DHODH Q02127 2/20 0.46
ALDH1A1 P00352 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29854461 0.86 MAPK14 (0.51) MKNK1CHEK2MKNK2PARP1BCAT2
SCHEMBL121338 0.85 ESR2 (0.58) ESR2HSD17B1L3MBTL1ALDH1A1RARB
SCHEMBL29707122 0.85 ESR2 (0.58) ESR2HSD17B1L3MBTL1ALDH1A1RARB
SCHEMBL9541786 0.85 PARP1 (0.52) HSD17B1PARP1L3MBTL1TSHRHSD17B10
SCHEMBL5608472 0.84 HSD17B1 (0.62) ESR2HSD17B1L3MBTL1MAPTALDH1A1
SCHEMBL3898821 0.84 PARP1 (0.48) MKNK1MKNK2PARP1L3MBTL1POLB
Hydrochloric Acid SCHEMBL5753140 0.84 ESR2 (0.56) ESR2HSD17B1L3MBTL1ALDH1A1RARB
SCHEMBL1787533 0.83 PARP1 (0.56) ESR2MKNK1MKNK2HSD17B1PARP1
SCHEMBL2026663 0.83 L3MBTL1 (0.52) MKNK1CHEK2MKNK2PARP1BCAT2
SCHEMBL30903715 0.83 L3MBTL1 (0.52) MKNK1CHEK2MKNK2PARP1BCAT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013028445-A1 FATTY ACID SYNTHASE INHIBITORS GLAXOSMITHKLINE LLC (US) 2013-02-28 WO claimed
CN-122029148-A N-phenyl-3- (2, 5-dioxopyrrolidin-1-yl) propionamide derivatives and similar compounds as DUX4 inhibitors for the treatment of, for example, neuromuscular diseases 阿勒泰治疗公司 2026-05-12 CN disclosed
US-20250179036-A1 MORPHOLINE-3-CARBOXAMIDE DERIVATIVES AS PROSTAGLANDIN E2 RECEPTOR 4 (EP4) AGONISTS FOR THE TREATMENT OF GASTROINTESTINAL AND PULMONARY DISEASES NXERA PHARMA UK LIMITED (GB) 2025-06-05 US disclosed
CN-104364246-B Piperidine derivatives useful as GPR119 agonists 株式会社钟根堂 2018-05-22 CN disclosed
CN-104470902-B N- (3-heteroarylaryl) -4-arylarylarylcarboxamides and analogs as Hedgehog pathway inhibitors and uses thereof 南京英派药业有限公司 2017-05-24 CN disclosed
EP-2681205-A1 BIARYL DERIVATIVES AS SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 2 INHIBITORS Universität des Saarlandes (DE) 2014-01-08 EP disclosed
WO-2013028445-A1 FATTY ACID SYNTHASE INHIBITORS GLAXOSMITHKLINE LLC (US) 2013-02-28 WO disclosed
WO-2012117097-A1 BIARYL DERIVATIVES AS SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 2 INHIBITORS Universität des Saarlandes (DE) 2012-09-07 WO disclosed
WO-2011075747-A1 THERAPEUTIC COMPOUNDS GLAXOSMITHKLINE LLC (US) 2011-06-23 WO disclosed
EP-2121621-A1 LXR AND FXR MODULATORS Exelixis, Inc. (US) 2009-11-25 EP disclosed
WO-2008073825-A1 LXR AND FXR MODULATORS EXELIXIS, INC. (US) 2008-06-19 WO disclosed
EP-0733048-A1 HETEROCYCLIC BIPHENYLYLAMIDES USEFUL AS 5HT1D ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1996-09-25 EP disclosed
WO-1995015954-A1 HETEROCYCLIC BIPHENYLYLAMIDES USEFUL AS 5HT1D ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1995-06-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250179036-A1 MORPHOLINE-3-CARBOXAMIDE DERIVATIVES AS PROSTAGLANDIN E2 RECEPTOR 4 (EP4) AGONISTS FOR THE TREATMENT OF GASTROINTESTINAL AND PULMONARY DISEASES PTGER4, PTGER1, PTGER2 ESR2 128/4885MKNK1 3311/4885CHEK2 3661/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.