SCHEMBL2027130

SCHEMBL2027130

O=c1[nH]c(=O)n(OCc2ccccc2)c2ncccc12

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LDHA P00338 1/20 0.45
HCAR2 Q8TDS4 7/20 0.44
SMN1; SMN2 Q16637 1/20 0.42
KDM4C Q9H3R0 1/20 0.41
PARP1 P09874 3/20 0.40
AURKA O14965 1/20 0.40
ELANE P08246 1/20 0.40
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
HPGD P15428 1/20 0.39
CYP2C19 P33261 1/20 0.39
ALDH1A1 P00352 1/20 0.39
TSHR P16473 1/20 0.39
KDM5C P41229 1/20 0.39
PNP P00491 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2027361 0.87 HCAR2 (0.48) HCAR2CYP1A2CYP2C9HPGDCYP2C19
SCHEMBL3515995 0.80 ALDH1A1 (0.44) SMN1; SMN2ELANEALDH1A1TSHR
SCHEMBL6731313 0.79 ALDH1A1 (0.50) SMN1; SMN2PARP1HPGDALDH1A1TSHR
SCHEMBL12640845 0.78 HPGD (0.44) LDHAHCAR2CYP1A2CYP2C9HPGD
SCHEMBL23234756 0.77 HPGD (0.48) LDHAPARP1AURKACYP1A2CYP2C9
SCHEMBL3514631 0.75 ALDH1A1 (0.41) LDHASMN1; SMN2ELANEALDH1A1TSHR
SCHEMBL3515379 0.75 KDM4E (0.45) SMN1; SMN2ELANECYP1A2ALDH1A1TSHR
SCHEMBL3517696 0.74 ALDH1A1 (0.40) SMN1; SMN2ELANECYP2C19ALDH1A1TSHR
SCHEMBL2023608 0.74 HPGD (0.45) LDHAHCAR2PARP1AURKACYP1A2
SCHEMBL3515597 0.73 ALDH1A1 (0.42) SMN1; SMN2KDM4CCYP2C9HPGDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011075747-A1 THERAPEUTIC COMPOUNDS GLAXOSMITHKLINE LLC (US) 2011-06-23 WO disclosed