SCHEMBL20301341

SCHEMBL20301341

CC1(C)N=C(c2nnc3c(F)c(F)ccc3n2)c2cccc(C(F)(F)F)c2C1(C)C

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 6/20 0.38
CYP1A2 P05177 4/20 0.33
CYP2D6 P10635 3/20 0.33
CLK4 Q9HAZ1 3/20 0.33
CYP2C19 P33261 3/20 0.33
CYP2C9 P11712 1/20 0.33
RECQL P46063 1/20 0.33
USP1 O94782 3/20 0.31
WDR48 Q8TAF3 3/20 0.31
CYP3A4 P08684 2/20 0.31
USP2 O75604 1/20 0.31
MEN1 O00255 1/20 0.31
TSHR P16473 1/20 0.31
KMT2A Q03164 1/20 0.31
HSD17B10 Q99714 1/20 0.31
MPL P40238 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20301006 0.90 HSD11B1 (0.37) HSD11B1CYP1A2CYP2D6CLK4CYP2C19
SCHEMBL20301138 0.89 HSD11B1 (0.37) HSD11B1CYP1A2CYP2D6CLK4CYP2C19
SCHEMBL20300999 0.89 HSD11B1 (0.31) HSD11B1
SCHEMBL20301404 0.87 MGAM (0.31) HSD11B1
SCHEMBL20300971 0.86 PDE2A (0.30)
SCHEMBL20300877 0.84
SCHEMBL20300902 0.82 HSD11B1 (0.34) HSD11B1CYP1A2CYP2D6CLK4CYP2C19
SCHEMBL20300883 0.81 HSD11B1 (0.33) HSD11B1CYP1A2CYP2D6CLK4CYP2C19
SCHEMBL20300899 0.81 PDE2A (0.31) HSD11B1
SCHEMBL20300863 0.80 HSD11B1 (0.38) HSD11B1MPL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018116072-A1 HETEROCYCLIC COMPOUNDS PI INDUSTRIES LTD. (IN) 2018-06-28 WO claimed
WO-2018116072-A1 HETEROCYCLIC COMPOUNDS PI INDUSTRIES LTD. (IN) 2018-06-28 WO disclosed