SCHEMBL20301375

SCHEMBL20301375

CC1(C)N=C(c2cc3ccccc3nn2)c2cccc(F)c2C1(F)F

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MBNL1 Q9NR56 1/20 0.38
NPC1 O15118 3/20 0.35
KDM4E B2RXH2 1/20 0.33
PDE10A Q9Y233 2/20 0.32
PDE2A O00408 1/20 0.32
BACE1 P56817 1/20 0.31
RPS6KA2 Q15349 1/20 0.31
ADORA2A P29274 1/20 0.30
ALDH1A1 P00352 1/20 0.30
MAPT P10636 1/20 0.30
RAB9A P51151 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20300767 0.89 KDM4E (0.31) MBNL1KDM4E
SCHEMBL20301236 0.89 MBNL1 (0.39) MBNL1NPC1KDM4EPDE10ARPS6KA2
SCHEMBL20300844 0.88 MBNL1 (0.35) MBNL1NPC1KDM4EPDE10AADORA2A
SCHEMBL20300689 0.88 NPC1 (0.35) MBNL1NPC1BACE1ALDH1A1MAPT
SCHEMBL20301186 0.88 KDM4E (0.36) MBNL1KDM4E
SCHEMBL20300735 0.86 KDM4E (0.33) KDM4E
SCHEMBL20300743 0.86 KDM4E (0.35) KDM4EPDE10APDE2AALDH1A1
SCHEMBL20301949 0.85 ACP1 (0.37) KDM4EBACE1
SCHEMBL20301394 0.85 KMT2A (0.35) MBNL1KDM4E
SCHEMBL20301474 0.82 NPC1 (0.40) MBNL1NPC1KDM4EPDE10AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018116072-A1 HETEROCYCLIC COMPOUNDS PI INDUSTRIES LTD. (IN) 2018-06-28 WO claimed
WO-2018116072-A1 HETEROCYCLIC COMPOUNDS PI INDUSTRIES LTD. (IN) 2018-06-28 WO disclosed