SCHEMBL20301474

SCHEMBL20301474

CC1(C)N=C(c2ccc3ccccc3n2)c2cccc(F)c2C1(F)F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.40
RAB9A P51151 6/20 0.40
SMN1; SMN2 Q16637 4/20 0.40
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
POLB P06746 2/20 0.40
LMNA P02545 2/20 0.40
PDE10A Q9Y233 2/20 0.39
AR P10275 10/20 0.39
PTGS2 P35354 1/20 0.39
MAPT P10636 3/20 0.38
ALDH1A1 P00352 3/20 0.38
CYP3A4 P08684 2/20 0.38
TP53 P04637 1/20 0.38
MAPK1 P28482 1/20 0.38
HIF1A Q16665 1/20 0.38
KDM4E B2RXH2 2/20 0.37
MBNL1 Q9NR56 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
CYP1A2 P05177 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15560843 0.88 PDE10A (0.40) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL20301261 0.86 AR (0.43) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL20300973 0.86 NPC1 (0.39) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL20300738 0.85 CNR2 (0.43) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL20301260 0.84 NPC1 (0.39) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL20301375 0.82 MBNL1 (0.38) NPC1RAB9ASMN1; SMN2PDE10AMAPT
SCHEMBL20300810 0.80 ADORA2A (0.35) MEN1KMT2APDE10AARMAPT
SCHEMBL20300854 0.79 AR (0.38) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL20301025 0.78 AR (0.45) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL20301266 0.77 ADORA2A (0.38) MEN1KMT2APDE10AARMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018116072-A1 HETEROCYCLIC COMPOUNDS PI INDUSTRIES LTD. (IN) 2018-06-28 WO claimed
WO-2018116072-A1 HETEROCYCLIC COMPOUNDS PI INDUSTRIES LTD. (IN) 2018-06-28 WO disclosed