SCHEMBL20304522

SCHEMBL20304522

CCOC(=O)CC(=O)c1ccc(C(C)(C)C)nc1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.43
KDM4E B2RXH2 2/20 0.43
ALDH1A1 P00352 2/20 0.43
MEN1 O00255 1/20 0.43
GAA P10253 3/20 0.43
MAPT P10636 6/20 0.42
NPC1 O15118 3/20 0.42
RAB9A P51151 3/20 0.42
SMN1; SMN2 Q16637 2/20 0.40
TSHR P16473 1/20 0.40
LMNA P02545 1/20 0.40
CXCR1 P25024 1/20 0.39
CXCR2 P25025 1/20 0.39
MGAM O43451 1/20 0.39
SI P14410 1/20 0.39
MGAM2 Q2M2H8 1/20 0.39
NPSR1 Q6W5P4 1/20 0.38
TP53 P04637 1/20 0.38
HPGD P15428 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10276146 0.87 NPC1 (0.46) KMT2AKDM4EALDH1A1MEN1GAA
SCHEMBL26315587 0.87 KMT2A (0.43) KMT2AKDM4EALDH1A1MEN1GAA
SCHEMBL10662120 0.82 HDAC1 (0.51) KMT2AKDM4EALDH1A1MEN1GAA
SCHEMBL29939457 0.82 HDAC1 (0.51) KMT2AKDM4EALDH1A1MEN1GAA
SCHEMBL12868073 0.82 KMT2A (0.54) KMT2AKDM4EMEN1GAAMAPT
SCHEMBL23149668 0.81 ALDH1A1 (0.47) KMT2AKDM4EALDH1A1MEN1GAA
SCHEMBL30786505 0.81 ALDH1A1 (0.47) KMT2AKDM4EALDH1A1MEN1GAA
SCHEMBL1474603 0.80 MAPT (0.42) KMT2AKDM4EMEN1MAPTNPC1
SCHEMBL3656932 0.79 KMT2A (0.46) KMT2AKDM4EALDH1A1MEN1GAA
SCHEMBL3173315 0.79 DGAT1 (0.60) KMT2AKDM4EALDH1A1MEN1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12358929-B2 NMDA receptor modulators and uses thereof NOVARTIS AG (CH) 2025-07-15 US disclosed
US-20240294546-A1 NMDA RECEPTOR MODULATORS AND USES THEREOF NOVARTIS AG (CH) 2024-09-05 US disclosed
EP-3558318-B1 NMDA RECEPTOR MODULATORS AND USES THEREOF NOVARTIS AG (CH) 2023-12-20 EP disclosed
US-11807650-B2 NMDA receptor modulators and uses thereof NOVARTIS AG (CH) 2023-11-07 US disclosed
US-11807650-B2 NMDA receptor modulators and uses thereof NOVARTIS AG (CH) 2023-11-07 US disclosed
US-11807650-B2 NMDA receptor modulators and uses thereof NOVARTIS AG (CH) 2023-11-07 US disclosed
US-20220153755-A1 NMDA RECEPTOR MODULATORS AND USES THEREOF NOVARTIS AG (CH) 2022-05-19 US disclosed
US-20220153755-A1 NMDA RECEPTOR MODULATORS AND USES THEREOF NOVARTIS AG (CH) 2022-05-19 US disclosed
US-11274107-B2 NMDA receptor modulators and uses thereof CADENT THERAPEUTICS, INC. (US) 2022-03-15 US disclosed
US-11274107-B2 NMDA receptor modulators and uses thereof CADENT THERAPEUTICS, INC. (US) 2022-03-15 US disclosed
US-20200087323-A1 NMDA RECEPTOR MODULATORS AND USES THEREOF NOVARTIS AG (CH) 2020-03-19 US disclosed
EP-3558318-A1 NMDA RECEPTOR MODULATORS AND USES THEREOF Cadent Therapeutics, Inc. (US) 2019-10-30 EP disclosed
WO-2018119374-A1 NMDA RECEPTOR MODULATORS AND USES THEREOF CADENT THERAPEUTICS (US) 2018-06-28 WO disclosed
WO-2018119374-A1 NMDA RECEPTOR MODULATORS AND USES THEREOF CADENT THERAPEUTICS (US) 2018-06-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11807650-B2 NMDA receptor modulators and uses thereof GRIN1, GRIN2A, GRIN2C KMT2A 602/4885KDM4E 1415/4885ALDH1A1 2036/4885
US-11274107-B2 NMDA receptor modulators and uses thereof GRIN1, GRIN2A, GRIN2C KMT2A 602/4885KDM4E 1415/4885ALDH1A1 2036/4885
US-20240294546-A1 NMDA RECEPTOR MODULATORS AND USES THEREOF GRIN1, GRIN2A, GRIN2C KMT2A 602/4885KDM4E 1415/4885ALDH1A1 2036/4885
US-12358929-B2 NMDA receptor modulators and uses thereof GRIN1, GRIN2A, GRIN2C KMT2A 602/4885KDM4E 1415/4885ALDH1A1 2036/4885
US-20200087323-A1 NMDA RECEPTOR MODULATORS AND USES THEREOF GRIN1, GRIN2A, GRIN2C KMT2A 602/4885KDM4E 1415/4885ALDH1A1 2036/4885
US-20220153755-A1 NMDA RECEPTOR MODULATORS AND USES THEREOF GRIN1, GRIN2A, GRIN2C KMT2A 602/4885KDM4E 1415/4885ALDH1A1 2036/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.