SCHEMBL20305409

SCHEMBL20305409

CCN(C(=O)c1cc2ccccc2[nH]1)[C@H]1CCC[C@@H](N(C)Cc2ccccc2)C1

nearest known ligand 0.57

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AR P10275 1/20 0.46
ATM Q13315 1/20 0.45
ACKR3 P25106 1/20 0.45
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
RXFP1 Q9HBX9 2/20 0.44
MDM2 Q00987 1/20 0.43
IDO1 P14902 1/20 0.43
ALDH1A1 P00352 1/20 0.43
CCKBR P32239 2/20 0.42
KDM4E B2RXH2 1/20 0.42
MAPT P10636 1/20 0.42
DAO P14920 1/20 0.42
HPGD P15428 1/20 0.42
SRD5A2 P31213 1/20 0.42
HSD17B10 Q99714 1/20 0.42
HDAC1 Q13547 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26346021 1.00 AR (0.46) ARATMACKR3MEN1KMT2A
SCHEMBL20320969 1.00 AR (0.46) ARATMACKR3MEN1KMT2A
SCHEMBL26009253 0.85 ATM (0.44) ATMMEN1KMT2ARXFP1IDO1
SCHEMBL27024206 0.83 KDM4E (0.45) ALDH1A1CCKBRKDM4EMAPTDAO
SCHEMBL8152104 0.83 CCKBR (0.52) MDM2ALDH1A1CCKBRKDM4EMAPT
SCHEMBL20305589 0.82 MDM2 (0.44) ARMDM2IDO1ALDH1A1CCKBR
SCHEMBL20320892 0.82 MDM2 (0.44) ARMDM2IDO1ALDH1A1CCKBR
SCHEMBL20320928 0.82 MDM2 (0.44) ARMDM2IDO1ALDH1A1CCKBR
SCHEMBL20320826 0.82 MDM2 (0.44) ARMDM2IDO1ALDH1A1CCKBR
SCHEMBL20320869 0.82 MDM2 (0.44) ARMDM2IDO1ALDH1A1CCKBR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4306166-A2 COMPOUNDS, COMPOSITIONS AND METHODS OF USE Aquinnah Pharmaceuticals Inc. (US) 2024-01-17 EP disclosed
US-20230303489-A1 COMPOUNDS, COMPOSITIONS AND METHODS OF USE AQUINNAH PHARMACEUTICALS INC (US) 2023-09-28 US disclosed
US-20230303489-A1 COMPOUNDS, COMPOSITIONS AND METHODS OF USE AQUINNAH PHARMACEUTICALS INC (US) 2023-09-28 US disclosed
EP-3557998-B1 COMPOUNS, COMPOSITIONS AND METHODS OF USE AQUINNAH PHARMACEUTICALS INC (US) 2023-08-16 EP disclosed
US-11542233-B2 Compounds, compositions and methods of use AQUINNAH PHARMACEUTICALS, INC. (US) 2023-01-03 US disclosed
US-11542233-B2 Compounds, compositions and methods of use AQUINNAH PHARMACEUTICALS, INC. (US) 2023-01-03 US disclosed
US-20200270211-A1 COMPOUNDS, COMPOSITIONS AND METHODS OF USE AQUINNAH PHARMACEUTICALS INC (US) 2020-08-27 US disclosed
US-20200270211-A1 COMPOUNDS, COMPOSITIONS AND METHODS OF USE AQUINNAH PHARMACEUTICALS INC (US) 2020-08-27 US disclosed
EP-3557998-A1 COMPOUNS, COMPOSITIONS AND METHODS OF USE Aquinnah Pharmaceuticals Inc. (US) 2019-10-30 EP disclosed
WO-2018119395-A1 COMPOUNS, COMPOSITIONS AND METHODS OF USE AQUINNAH PHARMACEUTICALS, INC. (US) 2018-06-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11542233-B2 Compounds, compositions and methods of use FUS, TFEB, CLN6 AR 4018/4885ATM 1839/4885ACKR3 4461/4885
US-20200270211-A1 COMPOUNDS, COMPOSITIONS AND METHODS OF USE FUS, TFEB, CLN6 AR 4018/4885ATM 1839/4885ACKR3 4461/4885
US-20230303489-A1 COMPOUNDS, COMPOSITIONS AND METHODS OF USE FUS, TFEB, CLN6 AR 4018/4885ATM 1839/4885ACKR3 4461/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.