SCHEMBL20312552

SCHEMBL20312552

CN(Cc1ccc(C#N)cc1)C(=O)c1cccc(CN2C(=N)NC(c3ccc(F)cc3)(c3ccc(F)cc3)C2=O)c1

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NSD2 O96028 2/20 0.52
KMT2A Q03164 3/20 0.44
ALDH1A1 P00352 1/20 0.42
HTT P42858 1/20 0.42
ROCK2 O75116 1/20 0.39
KCNH2 Q12809 1/20 0.39
MEN1 O00255 2/20 0.39
TACR3 P29371 2/20 0.38
HSD17B1 P14061 1/20 0.37
HSD17B2 P37059 1/20 0.37
KDM1A O60341 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20312651 0.93 ALDH1A1 (0.47) NSD2KMT2AALDH1A1HTTMEN1
SCHEMBL22344174 0.91 NSD2 (0.42) NSD2KMT2AALDH1A1HTTMEN1
SCHEMBL20312544 0.90 KMT2A (0.50) KMT2AALDH1A1HTTMEN1KDM1A
SCHEMBL22344170 0.89 ALDH1A1 (0.44) NSD2KMT2AALDH1A1HTTMEN1
SCHEMBL20303043 0.89 NSD2 (0.40) NSD2KMT2AALDH1A1HTTMEN1
SCHEMBL20302759 0.88 ALDH1A1 (0.42) KMT2AALDH1A1HTTMEN1HSD17B1
SCHEMBL20312631 0.86 NSD2 (0.46) NSD2KMT2AALDH1A1HTTROCK2
SCHEMBL22344147 0.86 ALDH1A1 (0.41) KMT2AALDH1A1HTTMEN1TACR3
SCHEMBL20302726 0.85 ALDH1A1 (0.42) KMT2AALDH1A1HTTMEN1
SCHEMBL20312681 0.84 ALDH1A1 (0.42) KMT2AALDH1A1HTTMEN1TACR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20200261421-A1 HETEROCYCLIC COMPOUNDS AS HIV PROTEASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2020-08-20 US disclosed
WO-2018118827-A1 HETEROCYCLIC COMPOUNDS AS HIV PROTEASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2018-06-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200261421-A1 HETEROCYCLIC COMPOUNDS AS HIV PROTEASE INHIBITORS PREP, SERPINB1, PEPD NSD2 1226/4885KMT2A 2246/4885ALDH1A1 1467/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.