SCHEMBL20329327

SCHEMBL20329327

CC[C@@H](C(=O)NC)N1C(=O)c2ccsc2C1=O

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GCK P35557 1/20 0.40
ALDH1A1 P00352 5/20 0.39
GAA P10253 5/20 0.36
NPSR1 Q6W5P4 3/20 0.36
TSHR P16473 1/20 0.34
LMNA P02545 1/20 0.32
HTT P42858 1/20 0.32
TP53 P04637 1/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
CES1 P23141 1/20 0.32
KDM4E B2RXH2 1/20 0.32
TAAR1 Q96RJ0 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16624015 0.71 CES1 (0.43) GCKALDH1A1GAANPSR1TSHR
SCHEMBL13574907 0.70 MEN1 (0.51) ALDH1A1GAATP53MEN1KMT2A
SCHEMBL13394194 0.66 ALDH1A1 (0.53) ALDH1A1GAANPSR1TSHRLMNA
SCHEMBL12601431 0.66 CYP1B1 (0.47) ALDH1A1GAANPSR1TSHRLMNA
SCHEMBL19370684 0.65 TP53 (0.49) ALDH1A1GAANPSR1LMNAHTT
SCHEMBL18366044 0.63 ALDH1A1 (0.47) ALDH1A1GAALMNAHTTTP53
SCHEMBL22698792 0.63 ALDH1A1 (0.47) ALDH1A1GAALMNAHTTTP53
SCHEMBL30587617 0.63 ALDH1A1 (0.47) ALDH1A1GAALMNAHTTTP53
SCHEMBL19658556 0.63 ALDH1A1 (0.47) ALDH1A1GAALMNAHTTTP53
SCHEMBL10391180 0.62 ALDH1A1 (0.55) GCKALDH1A1GAANPSR1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018118947-A1 THIENOPYRROLE DERIVATIVES FOR USE IN TARGETING PROTEINS, COMPOSITIONS, METHODS, AND USES THEREOF BIOTHERYX, INC. (US) 2018-06-28 WO disclosed