SCHEMBL20333136

SCHEMBL20333136

COC(=O)c1ccc(CN2C[C@@H](C)N(C(=O)OC(C)(C)C)C[C@@H]2C)cc1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.52
HDAC6 Q9UBN7 1/20 0.52
PDK1 Q15118 1/20 0.48
PDK2 Q15119 1/20 0.48
PDK3 Q15120 1/20 0.48
PDK4 Q16654 1/20 0.48
GPR119 Q8TDV5 1/20 0.43
MAPK14 Q16539 3/20 0.42
TBK1 Q9UHD2 1/20 0.42
KDM4E B2RXH2 1/20 0.41
SIRT1 Q96EB6 2/20 0.41
SIRT2 Q8IXJ6 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
LMNA P02545 1/20 0.40
TSHR P16473 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
CYP3A4 P08684 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15292045 0.87 PDK1 (0.51) PDK1PDK2PDK3PDK4GPR119
SCHEMBL4501274 0.86 PDK1 (0.53) PDK1PDK2PDK3PDK4GPR119
SCHEMBL107382 0.85 PDK1 (0.65) PDK1PDK2PDK3PDK4GPR119
SCHEMBL105646 0.85 PDK1 (0.65) PDK1PDK2PDK3PDK4GPR119
SCHEMBL105647 0.85 PDK1 (0.65) PDK1PDK2PDK3PDK4GPR119
SCHEMBL13810588 0.85 PDK1 (0.65) PDK1PDK2PDK3PDK4GPR119
SCHEMBL20333526 0.84 HDAC1 (0.53) HDAC1HDAC6GPR119KDM4EL3MBTL1
SCHEMBL28347328 0.84 HDAC1 (0.53) HDAC1HDAC6GPR119KDM4EL3MBTL1
SCHEMBL20304754 0.84 PDK1 (0.50) PDK1PDK2PDK3PDK4MAPK14
SCHEMBL28346940 0.84 HDAC1 (0.54) HDAC1HDAC6GPR119TBK1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110573497-A Histone deacetylase inhibitors 生物马林药物股份有限公司 2019-12-13 CN disclosed
WO-2018119362-A2 HISTONE DEACETYLASE INHIBITORS BIOMARIN PHARMACEUTICALS INC. (US) 2018-06-28 WO disclosed