SCHEMBL20344213

SCHEMBL20344213

Cc1nc2cc(Br)c(C=O)cc2[nH]1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.45
HSP90AA1 P07900 1/20 0.44
ESR2 Q92731 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
MAPT P10636 5/20 0.41
POLB P06746 4/20 0.41
KDM4E B2RXH2 4/20 0.41
HPGD P15428 3/20 0.41
RAB9A P51151 3/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
TYMS P04818 1/20 0.40
GAA P10253 2/20 0.40
HSD17B10 Q99714 1/20 0.40
PRKDC P78527 1/20 0.40
CHRNB2 P17787 1/20 0.39
CHRNA4 P43681 1/20 0.39
GRIA1 P42261 1/20 0.39
GRIA2 P42262 1/20 0.39
GRIA3 P42263 1/20 0.39
GRIA4 P48058 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5752591 0.80 ALDH1A1 (0.53) ALDH1A1HSP90AA1ESR2TDP1MAPT
SCHEMBL30065191 0.80 MAPT (0.50) ALDH1A1HSP90AA1ESR2TDP1MAPT
SCHEMBL28394278 0.80 MAPT (0.50) ALDH1A1HSP90AA1ESR2TDP1MAPT
SCHEMBL18288212 0.77 MAPT (0.47) ALDH1A1HSP90AA1ESR2TDP1MAPT
SCHEMBL29954905 0.77 ALDH1A1 (0.53) ALDH1A1HSP90AA1ESR2TDP1MAPT
SCHEMBL5752586 0.77 ALDH1A1 (0.53) ALDH1A1HSP90AA1ESR2TDP1MAPT
SCHEMBL855939 0.74 MAPT (0.49) ALDH1A1HSP90AA1ESR2TDP1MAPT
SCHEMBL13041691 0.73 ALDH1A1 (0.59) ALDH1A1HSP90AA1ESR2TDP1MAPT
SCHEMBL4230805 0.72 ALDH1A1 (0.56) ALDH1A1HSP90AA1ESR2TDP1MAPT
SCHEMBL17285612 0.72 HSP90AA1 (0.54) ALDH1A1HSP90AA1ESR2TDP1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3145930-B1 FUSED TRIAZOLE DERIVATIVES AS PHOSPHODIESTERASE 10A INHIBITORS Celon Pharma Sa (PL) 2018-07-04 EP disclosed