SCHEMBL20344652

SCHEMBL20344652

C=CCOc1cccc(C(=O)N=C)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.51
KAT6A Q92794 1/20 0.51
KDM4E B2RXH2 1/20 0.50
NPC1 O15118 1/20 0.50
RAB9A P51151 1/20 0.50
ADRB2 P07550 1/20 0.49
ADRB1 P08588 1/20 0.49
ADRB3 P13945 1/20 0.49
FFAR1 O14842 1/20 0.45
MAP1LC3B Q9GZQ8 1/20 0.45
MAP1LC3A Q9H492 1/20 0.45
GAA P10253 1/20 0.43
KMT2A Q03164 2/20 0.43
MEN1 O00255 1/20 0.43
LMNA P02545 1/20 0.43
MAPT P10636 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
MGLL Q99685 1/20 0.41
NR4A2 P43354 2/20 0.41
CHRNB2 P17787 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1668739 0.83 NPC1 (0.67) ALDH1A1KAT6AKDM4ENPC1RAB9A
SCHEMBL29784242 0.83 NPC1 (0.67) ALDH1A1KAT6AKDM4ENPC1RAB9A
SCHEMBL21157003 0.81 KMT2A (0.52) ALDH1A1KAT6AKDM4ENPC1RAB9A
SCHEMBL203644 0.81 PARP1 (0.56) ALDH1A1KAT6AKDM4ENPC1RAB9A
SCHEMBL5729029 0.81 ALDH1A1 (0.53) ALDH1A1KAT6AKDM4ENPC1RAB9A
SCHEMBL1092605 0.81 MAOB (0.59) ALDH1A1KDM4ENPC1RAB9AADRB2
SCHEMBL24653904 0.81 KAT6A (0.50) ALDH1A1KAT6AKDM4ENPC1RAB9A
SCHEMBL9739886 0.80 ALDH1A1 (0.52) ALDH1A1KAT6AKDM4ENPC1RAB9A
SCHEMBL27294341 0.80 ADRB2 (0.62) ALDH1A1KAT6AKDM4ENPC1RAB9A
SCHEMBL23748267 0.80 ALDH1A1 (0.58) ALDH1A1KAT6AKDM4ENPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3342771-A1 HETEROCYCLIC AMIDES AS KINASE INHIBITORS GlaxoSmithKline Intellectual Property Development Ltd (GB) 2018-07-04 EP disclosed