SCHEMBL20355296

SCHEMBL20355296

Cc1cccc(Nc2cc(N)nc(C)n2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.49
POLB P06746 2/20 0.48
NFKB1 P19838 1/20 0.47
MAPT P10636 5/20 0.47
TP53 P04637 4/20 0.47
LMNA P02545 2/20 0.47
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
SLC2A1 P11166 1/20 0.46
NOD1 Q9Y239 1/20 0.46
RXRA P19793 1/20 0.45
PPARG P37231 1/20 0.45
RXRG P48443 1/20 0.45
PPARD Q03181 1/20 0.45
PPARA Q07869 1/20 0.45
CYP1A2 P05177 1/20 0.44
CYP2D6 P10635 1/20 0.44
EGFR P00533 3/20 0.44
RECQL P46063 1/20 0.43
ADORA2A P29274 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15305716 0.87 RAB9A (0.55) NPSR1POLBNFKB1MAPTTP53
SCHEMBL11461593 0.85 CYP1A2 (0.60) NPSR1POLBMAPTTP53LMNA
SCHEMBL20354983 0.83 POLB (0.61) NPSR1POLBNFKB1MAPTTP53
SCHEMBL20355107 0.82 NPC1 (0.48) NPSR1POLBNFKB1MAPTTP53
SCHEMBL20355108 0.82 MAPT (0.66) POLBMAPTTP53NPC1RAB9A
SCHEMBL8798667 0.79 EGFR (0.61) NPSR1LMNARAB9AEGFR
SCHEMBL691393 0.79 ABCG2 (0.48) POLBMAPTLMNANPC1RAB9A
SCHEMBL20355745 0.77 CYP1A2 (0.73) NPSR1POLBNFKB1MAPTTP53
SCHEMBL29609757 0.76 NUDT1 (0.58) NPSR1POLBNFKB1MAPTTP53
SCHEMBL28736428 0.76 NUDT1 (0.58) NPSR1POLBNFKB1MAPTTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018122775-A1 HETEROARYL COMPOUNDS AND THEIR USE MINORYX THERAPEUTICS S.L. (ES) 2018-07-05 WO disclosed