SCHEMBL2035784

SCHEMBL2035784

CC(=O)c1cc(Cl)c2cccnc2c1N1CCC(NC(=O)C(C)C)C1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.43
RAB9A P51151 4/20 0.43
ALOX12 P18054 3/20 0.43
NCOA3 Q9Y6Q9 2/20 0.43
NCOA1 Q15788 1/20 0.43
HMOX1 P09601 1/20 0.43
HTR3E A5X5Y0 2/20 0.41
HTR3B O95264 2/20 0.41
HTR3A P46098 2/20 0.41
HTR3D Q70Z44 2/20 0.41
HTR3C Q8WXA8 2/20 0.41
L3MBTL1 Q9Y468 3/20 0.41
MTNR1A P48039 3/20 0.41
MTNR1B P49286 3/20 0.41
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
ALDH1A1 P00352 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2163699 1.00 NPC1 (0.43) NPC1RAB9AALOX12NCOA3NCOA1
SCHEMBL2017849 0.91 NPC1 (0.48) NPC1RAB9AALOX12NCOA3NCOA1
SCHEMBL2017854 0.91 NPC1 (0.48) NPC1RAB9AALOX12NCOA3NCOA1
SCHEMBL12403641 0.88 SMO (0.48) NPC1RAB9AALOX12NCOA3NCOA1
SCHEMBL2017031 0.87 NPC1 (0.48) NPC1RAB9AALOX12NCOA3NCOA1
SCHEMBL2017265 0.87 NPC1 (0.48) NPC1RAB9AALOX12NCOA3NCOA1
SCHEMBL2041986 0.86 NPC1 (0.43) NPC1RAB9AALOX12NCOA3NCOA1
SCHEMBL2017712 0.86 NPC1 (0.43) NPC1RAB9AALOX12NCOA3NCOA1
SCHEMBL2017715 0.85 MTNR1A (0.41) NPC1RAB9AALOX12NCOA3NCOA1
SCHEMBL2014007 0.84 SMO (0.51) NPC1RAB9AALOX12NCOA3NCOA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011075630-A1 SUBSTITUTED FUSED ARYL AND HETEROARYL DERIVATIVES AS PI3K INHIBITORS INCYTE CORPORATION (US) 2011-06-23 WO disclosed