SCHEMBL2017715

SCHEMBL2017715

CC(C)C(=O)NC1CCN(c2c(CCN)cc(Cl)c3cccnc23)C1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 3/20 0.41
MTNR1B P49286 3/20 0.41
L3MBTL1 Q9Y468 4/20 0.40
NPC1 O15118 5/20 0.39
RAB9A P51151 5/20 0.39
ALOX12 P18054 3/20 0.39
HMOX1 P09601 1/20 0.39
METAP2 P50579 2/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
NPSR1 Q6W5P4 2/20 0.38
NCOA1 Q15788 1/20 0.38
NCOA3 Q9Y6Q9 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
HTT P42858 2/20 0.38
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2013328 0.91 L3MBTL1 (0.45) L3MBTL1NPC1RAB9AALOX12METAP2
SCHEMBL2013778 0.89 NPC1 (0.44) MTNR1AMTNR1BL3MBTL1NPC1RAB9A
SCHEMBL2017712 0.86 NPC1 (0.43) MTNR1AMTNR1BL3MBTL1NPC1RAB9A
SCHEMBL2041986 0.86 NPC1 (0.43) MTNR1AMTNR1BL3MBTL1NPC1RAB9A
SCHEMBL2035784 0.85 NPC1 (0.43) MTNR1AMTNR1BL3MBTL1NPC1RAB9A
SCHEMBL2163699 0.85 NPC1 (0.43) MTNR1AMTNR1BL3MBTL1NPC1RAB9A
SCHEMBL2012926 0.85 SMO (0.48) L3MBTL1NPC1RAB9AALOX12METAP2
SCHEMBL2018209 0.84 BTK (0.36) MTNR1AMTNR1BL3MBTL1NPC1RAB9A
SCHEMBL2011476 0.82 METAP2 (0.43) L3MBTL1NPC1RAB9AALOX12METAP2
SCHEMBL2011479 0.82 METAP2 (0.43) L3MBTL1NPC1RAB9AALOX12METAP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011075630-A1 SUBSTITUTED FUSED ARYL AND HETEROARYL DERIVATIVES AS PI3K INHIBITORS INCYTE CORPORATION (US) 2011-06-23 WO disclosed