SCHEMBL2036464

SCHEMBL2036464

O=C(NCc1ccccc1)c1ccc2c(c1)OCCN2

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.69
RAB9A P51151 2/20 0.69
HSD17B10 Q99714 1/20 0.69
PRMT5 O14744 1/20 0.54
WDR77 Q9BQA1 1/20 0.54
NPC1 O15118 3/20 0.53
KLF5 Q13887 2/20 0.53
ALDH1A1 P00352 4/20 0.53
MAPT P10636 2/20 0.53
KDM4E B2RXH2 1/20 0.53
ROCK2 O75116 1/20 0.52
ROCK1 Q13464 1/20 0.52
PKM P14618 1/20 0.51
PAX8 Q06710 1/20 0.51
ALOX12 P18054 1/20 0.49
ADORA3 P0DMS8 1/20 0.49
ADORA2A P29274 1/20 0.49
ADORA2B P29275 1/20 0.49
ADORA1 P30542 1/20 0.49
TSHR P16473 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19859136 0.84 EPHX2 (0.52) HPGDRAB9AHSD17B10PRMT5WDR77
SCHEMBL19864681 0.83 RAB9A (0.48) HPGDRAB9AHSD17B10PRMT5WDR77
SCHEMBL22145584 0.82 RAB9A (1.00) HPGDRAB9AHSD17B10NPC1KLF5
SCHEMBL14072996 0.80 TSHR (0.61) HPGDRAB9AHSD17B10PRMT5WDR77
SCHEMBL6981710 0.79 KDM4E (0.60) HPGDRAB9AHSD17B10NPC1ALDH1A1
SCHEMBL19260062 0.79 RAB9A (0.52) HPGDRAB9AHSD17B10NPC1ALDH1A1
SCHEMBL29566033 0.77 MAPT (0.55) RAB9AHSD17B10PRMT5WDR77NPC1
SCHEMBL4290086 0.77 MAPT (0.55) RAB9AHSD17B10PRMT5WDR77NPC1
SCHEMBL647939 0.77 RAB9A (0.84) HPGDRAB9AHSD17B10NPC1KLF5
SCHEMBL18280561 0.76 ROCK2 (0.53) PRMT5WDR77NPC1ALDH1A1ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011073276-A1 BENZOXAZINE ARYL SULFONAMIDE DERIVATIVES AS KV1.3 MODULATORS EVOTEC AG (DE) 2011-06-23 WO disclosed