SCHEMBL2036865

SCHEMBL2036865

COc1cc(F)c(-c2c(OC)nnc(C)c2-c2c(F)nc(C)c(F)c2F)c(F)c1

nearest known ligand 0.37

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GRM8 O00222 1/20 0.37
CYP1A2 P05177 1/20 0.37
GRM7 Q14831 1/20 0.37
PDE2A O00408 3/20 0.32
PDE10A Q9Y233 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3331310 0.74 RAC1 (0.39) GRM8CYP1A2GRM7PDE2APDE10A
SCHEMBL12394014 0.74 MEN1 (0.49) GRM8CYP1A2GRM7PDE2APDE10A
SCHEMBL1162395 0.72 CYP1A2 (0.41) GRM8CYP1A2GRM7PDE2APDE10A
SCHEMBL3611240 0.72 NPC1 (0.38) CYP1A2PDE2APDE10A
SCHEMBL2321107 0.71 ERN1 (0.39) CYP1A2
SCHEMBL2319119 0.71 GRM8 (0.33) GRM8CYP1A2GRM7PDE2APDE10A
SCHEMBL1872289 0.70 NPC1 (0.37) GRM8CYP1A2GRM7PDE2APDE10A
SCHEMBL2036866 0.69 PDE2A (0.40) GRM8CYP1A2GRM7PDE2APDE10A
SCHEMBL2318886 0.68 PIK3CD (0.34) GRM8CYP1A2GRM7PDE2APDE10A
SCHEMBL25356232 0.67 TAAR1 (0.47) GRM8CYP1A2GRM7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011076501-A1 NOVEL 5-(PYRIDIN-3-YL)-PYRIDANIZE DERIVATIVES AND THEIR USE AS MICROBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2011-06-30 WO disclosed