SCHEMBL203886

SCHEMBL203886

Fc1ccc(Nc2ccc(CNC3CC3)cc2)c(C(F)(F)F)c1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 3/20 0.41
CNR1 P21554 2/20 0.41
CCR3 P51677 1/20 0.40
BCHE P06276 3/20 0.40
ACHE P22303 3/20 0.40
BACE1 P56817 3/20 0.40
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
RAB9A P51151 1/20 0.38
CHEK1 O14757 1/20 0.38
HRH3 Q9Y5N1 1/20 0.37
CYP2D6 P10635 1/20 0.36
KCNH2 Q12809 1/20 0.36
GRIN2B Q13224 1/20 0.36
TEAD1 P28347 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL186185 0.78 LOXL2 (0.44) CNR2CNR1MEN1KMT2A
SCHEMBL185133 0.74 CNR2 (0.41) CNR2CNR1RAB9A
SCHEMBL19418435 0.74 MAPK10 (0.47) CNR2
SCHEMBL13159687 0.74 MAPK10 (0.47) CNR2
SCHEMBL1239998 0.73 BCHE (0.61) CCR3BCHEACHEBACE1MEN1
SCHEMBL184742 0.72 CYP3A4 (0.40) CNR2CNR1RAB9A
SCHEMBL5556152 0.69 BCHE (0.64) BCHEACHEBACE1MEN1KMT2A
SCHEMBL10073807 0.68 MEN1 (0.69) BCHEACHEBACE1MEN1KMT2A
SCHEMBL23124775 0.68 MEN1 (0.41) BCHEACHEBACE1MEN1KMT2A
Hydrochloric Acid SCHEMBL218521 0.68 BCHE (0.62) BCHEACHEBACE1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401256-A1 COMPOUNDS AS BRADYKININ B1 ANTAGONISTS Boehringer Ingelheim International GmbH (DE) 2012-01-04 EP disclosed
WO-2010097372-A1 COMPOUNDS AS BRADYKININ B1 ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-02 WO disclosed