SCHEMBL20405702

SCHEMBL20405702

COC(=O)c1cccc(C2=NBC(c3nnn(-c4ccccc4F)c3-c3ccccc3)=N2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 1/20 0.44
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
ALDH1A1 P00352 2/20 0.40
NPSR1 Q6W5P4 1/20 0.40
GABRG2 P18507 1/20 0.39
GABRB3 P28472 1/20 0.39
GABRA5 P31644 1/20 0.39
GABRA3 P34903 1/20 0.39
GRM5 P41594 2/20 0.37
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
NEK1 Q96PY6 1/20 0.36
AXL P30530 1/20 0.36
ERN1 O75460 1/20 0.36
IL2 P60568 1/20 0.36
IDO1 P14902 1/20 0.35
TDO2 P48775 1/20 0.35
GPR84 Q9NQS5 2/20 0.35
ACLY P53396 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3760933 0.79 NPC1 (0.62) DHODHNPC1RAB9AALDH1A1NPSR1
SCHEMBL3455957 0.73 NPC1 (0.50) DHODHNPC1RAB9AALDH1A1NPSR1
SCHEMBL3468631 0.72 MAPT (0.50) NPC1RAB9AALDH1A1NPSR1KMT2A
SCHEMBL3456402 0.69 NPC1 (0.48) NPC1RAB9AALDH1A1NPSR1
SCHEMBL13765570 0.66 MEN1 (0.47) ALDH1A1NPSR1KMT2AMEN1
SCHEMBL3753122 0.64 ALDH1A1 (0.56) ALDH1A1NPSR1KDM4ESMN1; SMN2
SCHEMBL7824107 0.64 RAB9A (0.68) NPC1RAB9AALDH1A1GABRG2GABRB3
SCHEMBL1221576 0.63 TSHR (0.67) RAB9AGABRG2GABRB3GABRA5GABRA3
SCHEMBL29410906 0.63 TSHR (0.67) RAB9AGABRG2GABRB3GABRA5GABRA3
SCHEMBL20162908 0.62 GAA (0.51) ALDH1A1NPSR1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2250165-B1 TRIAZOLE OXADIAZOLES DERIVATIVES MERCK SERONO SA (CH) 2018-07-25 EP disclosed