SCHEMBL2040686

SCHEMBL2040686

COc1cc(F)c(-c2c(Cl)nnc(C)c2-c2ccc(C(F)F)nc2)c(F)c1

nearest known ligand 0.33

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CTSA P10619 1/20 0.33
HDAC6 Q9UBN7 1/20 0.32
SLC34A1 Q06495 2/20 0.32
PDE2A O00408 1/20 0.31
PDE10A Q9Y233 1/20 0.31
GRM8 O00222 1/20 0.31
CYP1A2 P05177 1/20 0.31
GRM7 Q14831 1/20 0.31
PTGES O14684 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2032613 0.89 SLC34A1 (0.36) SLC34A1PTGES
SCHEMBL1873473 0.86 NPC1 (0.37) CTSAPDE2APDE10AGRM8CYP1A2
SCHEMBL2034115 0.82 PDE10A (0.39) PDE10AGRM8CYP1A2GRM7
SCHEMBL2320981 0.81 CTSA (0.31) CTSAPDE2APDE10AGRM8CYP1A2
SCHEMBL2354029 0.81 MEN1 (0.43) GRM8CYP1A2GRM7
SCHEMBL2318082 0.81 CTSA (0.32) CTSAPDE2APDE10A
SCHEMBL2039642 0.80 SLC34A1 (0.32) SLC34A1
SCHEMBL1162374 0.79 CYP1A2 (0.37) CTSAPDE2APDE10AGRM8CYP1A2
SCHEMBL2322215 0.79 BACE1 (0.35)
SCHEMBL2347440 0.76 NPC1 (0.39) CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011076501-A1 NOVEL 5-(PYRIDIN-3-YL)-PYRIDANIZE DERIVATIVES AND THEIR USE AS MICROBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2011-06-30 WO claimed
WO-2011076501-A1 NOVEL 5-(PYRIDIN-3-YL)-PYRIDANIZE DERIVATIVES AND THEIR USE AS MICROBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2011-06-30 WO disclosed