SCHEMBL2318082

SCHEMBL2318082

COc1cc(F)c(-c2c(Cl)nnc(C)c2-c2ccc(C#CCl)nc2)c(F)c1

nearest known ligand 0.32

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CTSA P10619 1/20 0.32
PDE2A O00408 1/20 0.32
PDE10A Q9Y233 1/20 0.32
GRM5 P41594 1/20 0.31
MCHR1 Q99705 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2322215 0.90 BACE1 (0.35) GRM5MCHR1
SCHEMBL2318504 0.89 PTGES (0.31)
SCHEMBL2320981 0.88 CTSA (0.31) CTSAPDE2APDE10A
SCHEMBL2322837 0.84 PDE2A (0.32) CTSAPDE2APDE10A
SCHEMBL1873473 0.84 NPC1 (0.37) CTSAPDE2APDE10A
SCHEMBL2040686 0.81 CTSA (0.33) CTSAPDE2APDE10A
SCHEMBL2034115 0.81 PDE10A (0.39) PDE10A
SCHEMBL2354029 0.79 MEN1 (0.43)
SCHEMBL1162374 0.78 CYP1A2 (0.37) CTSAPDE2APDE10A
SCHEMBL2319994 0.77 GABRA1 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011095459-A1 PYRIDAZINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR USE AS FUNGICIDES SYNGENTA PARTICIPATIONS AG (CH) 2011-08-11 WO claimed
WO-2011095459-A1 PYRIDAZINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR USE AS FUNGICIDES SYNGENTA PARTICIPATIONS AG (CH) 2011-08-11 WO disclosed