SCHEMBL20428554

SCHEMBL20428554

CCCOCn1nc(-c2ccc(Br)cc2)nc1OCC

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 3/20 0.45
NR1H3 Q13133 3/20 0.45
DGAT1 O75907 4/20 0.43
ADORA3 P0DMS8 5/20 0.38
ADORA2A P29274 2/20 0.38
AHR P35869 4/20 0.35
TP53 P04637 1/20 0.34
MAPT P10636 1/20 0.34
RARB P10826 1/20 0.33
GAA P10253 1/20 0.33
ADORA1 P30542 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16661015 0.89 DGAT1 (0.56) NR1H2NR1H3DGAT1ADORA3ADORA2A
SCHEMBL16661188 0.88 NR1H2 (0.41) NR1H2NR1H3DGAT1ADORA3ADORA2A
SCHEMBL16660978 0.75 DGAT1 (0.74) NR1H2NR1H3DGAT1AHRTP53
SCHEMBL21064877 0.74 DGAT1 (0.56) NR1H2NR1H3DGAT1AHRTP53
SCHEMBL16660852 0.73 DGAT1 (0.50) NR1H2NR1H3DGAT1AHRTP53
SCHEMBL16660890 0.73 DGAT1 (0.80) DGAT1
SCHEMBL16787869 0.72 DGAT1 (0.62) NR1H2NR1H3DGAT1ADORA2A
SCHEMBL16660877 0.72 DGAT1 (0.61) DGAT1MAPT
SCHEMBL16661342 0.67 DGAT1 (0.44) NR1H2NR1H3DGAT1AHRTP53
SCHEMBL16660927 0.66 DGAT1 (0.53) NR1H2NR1H3DGAT1AHRTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2862856-B1 IMIDAZOLE AND TRIAZOLE COMPOUNDS AS DGAT-1 INHIBITORS MITSUBISHI TANABE PHARMA CORP (JP) 2018-08-01 EP disclosed