SCHEMBL20432151

SCHEMBL20432151

CCCn1c(=O)n(CCCO)c(=O)c2c1nc(Cl)n2Cl

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 9/20 0.50
ADORA2A P29274 8/20 0.50
PDE4A P27815 4/20 0.50
PDE4B Q07343 4/20 0.50
PDE4C Q08493 4/20 0.50
PDE4D Q08499 4/20 0.50
CYP1A2 P05177 2/20 0.45
CYP2C19 P33261 1/20 0.45
RECQL P46063 1/20 0.45
CYP3A4 P08684 1/20 0.43
BLM P54132 1/20 0.43
PMP22 Q01453 1/20 0.43
HSD17B10 Q99714 1/20 0.43
ADORA3 P0DMS8 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL836600 0.83 CYP1A2 (0.47) ADORA2BADORA2APDE4APDE4BPDE4C
SCHEMBL16028356 0.80 TRPC5 (0.54) ADORA2BADORA2APDE4APDE4BPDE4C
SCHEMBL836842 0.78 CYP1A2 (0.53) ADORA2BADORA2APDE4APDE4BPDE4C
SCHEMBL16027932 0.75 CYP1A2 (0.44) ADORA2BADORA2APDE4APDE4BPDE4C
SCHEMBL3115778 0.74 CYP1A2 (0.52) ADORA2BADORA2APDE4APDE4BPDE4C
SCHEMBL16028494 0.72 ADORA3 (0.58) ADORA2BADORA2AADORA3
SCHEMBL16028059 0.72 TRPC5 (0.54) CYP1A2CYP2C19CYP3A4ADORA3
SCHEMBL16028583 0.71 TRPC5 (0.59) ADORA2BADORA2APDE4APDE4BPDE4C
SCHEMBL16027836 0.71 PCSK9 (0.48) CYP1A2CYP2C19CYP3A4ADORA3
SCHEMBL9430619 0.69 ADORA2A (0.61) ADORA2BADORA2APDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970303-B3 SUBSTITUTED XANTHINES AND METHODS OF USE THEREOF HYDRA BIOSCIENCES INC (US) 2018-08-01 EP disclosed