SCHEMBL20437623

SCHEMBL20437623

COc1nc(C)cc(N2CC3CC2CO3)n1

nearest known ligand 0.45

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MAP3K12 Q12852 17/20 0.45
DLK1 P80370 1/20 0.45
LRRK2 Q5S007 1/20 0.43
KCNQ3 O43525 1/20 0.41
KCNQ2 O43526 1/20 0.41
MAP3K13 O43283 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20437512 0.88 MAP3K12 (0.36) MAP3K12DLK1LRRK2MAP3K13
SCHEMBL22723429 0.86 MAP3K12 (0.44) MAP3K12DLK1LRRK2MAP3K13
SCHEMBL22723567 0.86 MAP3K12 (0.44) MAP3K12DLK1LRRK2MAP3K13
SCHEMBL22753142 0.86 MAP3K12 (0.44) MAP3K12DLK1LRRK2MAP3K13
SCHEMBL20437482 0.83 MAP3K12 (0.48) MAP3K12DLK1MAP3K13
SCHEMBL20437510 0.74 MAP3K12 (0.35) MAP3K12DLK1LRRK2MAP3K13
SCHEMBL20438009 0.73 HRH3 (0.42) LRRK2
SCHEMBL22723456 0.73 MAP3K12 (0.46) MAP3K12DLK1MAP3K13
SCHEMBL22723461 0.73 MAP3K12 (0.46) MAP3K12DLK1MAP3K13
SCHEMBL22753144 0.73 MAP3K12 (0.46) MAP3K12DLK1MAP3K13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018137593-A1 COMPOUNDS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2018-08-02 WO disclosed