SCHEMBL20439382

SCHEMBL20439382

c1ccc(COc2ccc([C@@H]3COc4cc5c(cnn5C5CCCCO5)cc4N3)cc2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 3/20 0.41
CYP4A11 Q02928 3/20 0.41
RXRA P19793 1/20 0.41
RXRB P28702 1/20 0.41
RXRG P48443 1/20 0.41
ATR Q13535 1/20 0.37
MCHR1 Q99705 6/20 0.36
KCNH2 Q12809 4/20 0.36
MMP13 P45452 1/20 0.34
USP2 O75604 1/20 0.34
GLA P06280 1/20 0.34
HTT P42858 1/20 0.34
EGFR P00533 1/20 0.34
MCHR2 Q969V1 1/20 0.34
NPC1 O15118 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
NFKB1 P19838 1/20 0.33
MAOB P27338 1/20 0.33
GRM5 P41594 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL680099 0.75 RXRA (0.49) CYP4F2CYP4A11RXRARXRBRXRG
SCHEMBL20439364 0.74 MAOB (0.42) KCNH2NPC1ALDH1A1HPGDNFKB1
SCHEMBL20439440 0.73 CYP4F2 (0.40) CYP4F2CYP4A11RXRARXRBRXRG
SCHEMBL5357173 0.73 MAOB (0.51) KCNH2MMP13NPC1ALDH1A1HPGD
SCHEMBL5357169 0.73 MAOB (0.51) KCNH2MMP13NPC1ALDH1A1HPGD
SCHEMBL20439439 0.72 CYP4F2 (0.41) CYP4F2CYP4A11RXRARXRBRXRG
SCHEMBL1366880 0.72 CYP4F2 (0.51) CYP4F2CYP4A11RXRARXRBRXRG
SCHEMBL30707091 0.71 RXRA (0.54) CYP4F2CYP4A11RXRARXRBRXRG
SCHEMBL20398080 0.71 RXRA (0.59) CYP4F2CYP4A11RXRARXRBRXRG
SCHEMBL25417935 0.71 RXRA (0.46) CYP4F2CYP4A11RXRARXRBRXRG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018138739-A1 NOVEL ANTIESTROGENIC HETEROCYCLIC COMPOUNDS SUN PHARMA ADVANCED RESEARCH COMPANY LIMITED (IN) 2018-08-02 WO disclosed