SCHEMBL20443302

SCHEMBL20443302

Cc1cc(-c2cc(C=O)ccc2Oc2ccc(Br)cc2F)c2cc[nH]c2n1

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 7/20 0.41
MET P08581 7/20 0.40
ROCK2 O75116 2/20 0.40
KDR P35968 1/20 0.40
FLT3 P36888 1/20 0.40
TRPA1 O75762 1/20 0.36
CCNK O75909 1/20 0.36
CDK12 Q9NYV4 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.35
JAK1 P23458 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20442999 0.85 ROCK2 (0.46) BRD4METROCK2KDRFLT3
SCHEMBL28643992 0.85 ROCK2 (0.43) BRD4METROCK2KDRFLT3
SCHEMBL20443319 0.83 ROCK2 (0.40) BRD4METROCK2KDRFLT3
SCHEMBL20443239 0.83 S1PR4 (0.41) BRD4METROCK2TRPA1CCNK
SCHEMBL20443297 0.82 ROCK2 (0.40) BRD4METROCK2KDRFLT3
SCHEMBL20443013 0.81 ROCK2 (0.39) BRD4METROCK2KDRFLT3
SCHEMBL20442994 0.81 BRD4 (0.53) BRD4
SCHEMBL20442995 0.79 ROCK2 (0.41) BRD4METROCK2KDRFLT3
SCHEMBL20443032 0.78 ROCK2 (0.40) BRD4METROCK2KDRFLT3
SCHEMBL20442964 0.78 BRD4 (0.47) BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110198941-B Pyrrolopyridine N-oxide derivative and preparation method and application thereof 江苏豪森药业集团有限公司 2021-09-28 CN disclosed
WO-2018137655-A1 PYRROLO-PYRIDINES N-OXIDE DERIVATIVE, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF 江苏豪森药业集团有限公司 2018-08-02 WO disclosed