SCHEMBL20443239

SCHEMBL20443239

Cc1cc(-c2cc([N+](=O)[O-])ccc2Oc2ccc(Br)cc2F)c2cc[nH]c2n1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
S1PR4 O95977 3/20 0.41
BRD4 O60885 1/20 0.39
AMY1A P0DUB6 1/20 0.39
HSPB1 P04792 4/20 0.39
ROCK2 O75116 1/20 0.39
MET P08581 1/20 0.36
LMNA P02545 1/20 0.36
KMT2A Q03164 1/20 0.36
TRPA1 O75762 1/20 0.35
CCNK O75909 1/20 0.35
CDK12 Q9NYV4 1/20 0.35
HTT P42858 1/20 0.34
ALDH1A1 P00352 1/20 0.34
TTBK1 Q5TCY1 1/20 0.34
TTBK2 Q6IQ55 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
SCN9A Q15858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20442999 0.83 ROCK2 (0.46) BRD4ROCK2METTRPA1CCNK
SCHEMBL28643992 0.83 ROCK2 (0.43) BRD4ROCK2METTRPA1CCNK
SCHEMBL20443302 0.83 BRD4 (0.41) BRD4ROCK2METTRPA1CCNK
SCHEMBL20443319 0.82 ROCK2 (0.40) BRD4ROCK2METTRPA1CCNK
SCHEMBL20443297 0.81 ROCK2 (0.40) BRD4ROCK2METTRPA1CCNK
SCHEMBL29548670 0.81 HSPB1 (0.45) S1PR4AMY1AHSPB1LMNAKMT2A
SCHEMBL28721761 0.81 HSPB1 (0.45) S1PR4AMY1AHSPB1LMNAKMT2A
SCHEMBL20443013 0.79 ROCK2 (0.39) BRD4ROCK2METTRPA1CCNK
SCHEMBL20442994 0.79 BRD4 (0.53) BRD4
SCHEMBL20442995 0.78 ROCK2 (0.41) BRD4ROCK2METTRPA1CCNK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110198941-B Pyrrolopyridine N-oxide derivative and preparation method and application thereof 江苏豪森药业集团有限公司 2021-09-28 CN disclosed
WO-2018137655-A1 PYRROLO-PYRIDINES N-OXIDE DERIVATIVE, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF 江苏豪森药业集团有限公司 2018-08-02 WO disclosed