SCHEMBL2044752

SCHEMBL2044752

CC(=O)c1ccccc1-c1nc(C(=N)N(C#N)C2CCCCCCC2)cs1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.37
SLC6A9 P48067 1/20 0.35
SLC6A5 Q9Y345 1/20 0.35
ACHE P22303 3/20 0.34
TYR P14679 1/20 0.34
HTR2B P41595 1/20 0.33
EIF4E P06730 1/20 0.33
MAOA P21397 1/20 0.33
HTR2C P28335 2/20 0.32
HPGD P15428 1/20 0.32
TSHR P16473 1/20 0.32
UCHL1 P09936 1/20 0.32
USP30 Q70CQ3 1/20 0.32
PIN1 Q13526 1/20 0.32
CHRM1 P11229 1/20 0.32
KDM4E B2RXH2 2/20 0.32
SPHK1 Q9NYA1 2/20 0.32
ALDH1A1 P00352 1/20 0.32
APAF1 O14727 1/20 0.32
NPC1 O15118 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3547753 0.78 SLC6A9 (0.44) HRH3SLC6A9SLC6A5TSHRKDM4E
SCHEMBL4973482 0.75 SLC6A9 (0.42) HRH3SLC6A9SLC6A5HPGDTSHR
SCHEMBL2027225 0.73 TYR (0.61) TYRHPGDPIN1KDM4EALDH1A1
SCHEMBL3543022 0.73 TYR (0.61) TYRHPGDPIN1KDM4EALDH1A1
SCHEMBL2026846 0.73 PDE4D (0.38) HRH3ACHETYRHTR2BEIF4E
SCHEMBL2026844 0.73 TYR (0.44) HRH3TYRHPGDPIN1KDM4E
SCHEMBL2026842 0.73 TYR (0.44) HRH3TYRHPGDPIN1KDM4E
SCHEMBL5662015 0.71 HTT (0.46) HRH3ACHEHTR2BHTR2CHPGD
SCHEMBL3536540 0.70 CNR1 (0.45) HRH3HTR2CNPC1RAB9A
SCHEMBL3537686 0.70 ACHE (0.62) ACHEHTR2BEIF4EMAOAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2243479-A2 Novel amide and amidine derivates and uses thereof Abbott Laboratories (US) 2010-10-27 EP claimed
WO-2011068927-A2 11-β-HYDROXYSTEROID DEHYDROGENASE TYPE 1 (11B-HSD1) INHIBITORS AND USES THEREOF ABBOTT LABORATORIES (US) 2011-06-09 WO disclosed