SCHEMBL20448229

SCHEMBL20448229

Cc1[c]c(OCC(F)(F)C(F)F)c(C)cc1

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.37
ALDH1A1 P00352 2/20 0.37
LMNA P02545 1/20 0.37
CFTR P13569 4/20 0.35
POLB P06746 1/20 0.33
GAA P10253 1/20 0.33
KMT2A Q03164 2/20 0.32
MEN1 O00255 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
HTT P42858 2/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20135752 0.83 CNR2 (0.33) ALDH1A1KMT2AMEN1SMN1; SMN2
SCHEMBL20916973 0.76
SCHEMBL17815773 0.69 SMN1; SMN2 (0.41) MAPK1ALDH1A1LMNAPOLBGAA
SCHEMBL1710086 0.68 KDM4E (0.45) ALDH1A1LMNACFTRKMT2AMEN1
SCHEMBL1710061 0.67 KMT2A (0.51) MAPK1ALDH1A1CFTRPOLBGAA
SCHEMBL20135751 0.67
SCHEMBL17247992 0.65 MAPK1 (0.43) MAPK1ALDH1A1LMNACFTR
SCHEMBL5982679 0.65 ALDH1A1 (0.36) ALDH1A1LMNACFTRKMT2AMEN1
SCHEMBL5430591 0.63 HTT (0.43) MAPK1ALDH1A1CFTRPOLBGAA
SCHEMBL17811834 0.62 HTT (0.37) MAPK1ALDH1A1LMNAKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 37 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4139304-A1 2-(HET)ARYL-SUBSTITUTED CONDENSED HETEROCYCLIC DERIVATIVES AS PEST CONTROL AGENTS Bayer Aktiengesellschaft (DE) 2023-03-01 EP disclosed
EP-4003966-A1 5-AMINO SUBSTITUTED PYRAZOLES AND TRIAZOLES AS PEST CONTROL AGENTS Bayer Aktiengesellschaft (DE) 2022-06-01 EP disclosed
EP-3993626-A1 HERBICIDAL COMPOSITIONS Bayer Aktiengesellschaft (DE) 2022-05-11 EP disclosed
EP-3982732-A1 STABILIZED DITHIOCARBAMATE FORMULATIONS Bayer Aktiengesellschaft (DE) 2022-04-20 EP disclosed
WO-2021213978-A1 2-(HET)ARYL-SUBSTITUTED CONDENSED HETEROCYCLIC DERIVATIVES AS PEST CONTROL AGENTS BAYER AKTIENGESELLSCHAFT (DE) 2021-10-28 WO disclosed
EP-3515921-B1 PYRAZOLO[1,5-A]PYRIDINE DERIVATIVES AND THEIR USE AS PESTICIDES BAYER CROPSCIENCE AG (DE) 2021-10-27 EP disclosed
EP-3849975-A1 HETEROCYCLENE DERIVATIVES AS PEST CONTROL AGENTS Bayer Aktiengesellschaft (DE) 2021-07-21 EP disclosed
EP-3814346-A1 HETEROCYCLENE DERIVATIVES AS PEST CONTROL AGENTS Bayer Aktiengesellschaft (DE) 2021-05-05 EP disclosed
EP-3772960-A1 ACTIVE INGREDIENT COMBINATIONS WITH INSECTICIDAL, FUNGICIDAL AND ACARICIDAL PROPERTIES Bayer Aktiengesellschaft (DE) 2021-02-17 EP disclosed
WO-2021013721-A1 5-AMINO SUBSTITUTED PYRAZOLES AND TRIAZOLES AS PEST CONTROL AGENTS BAYER AKTIENGESELLSCHAFT (DE) 2021-01-28 WO disclosed
WO-2019162174-A1 CONDENSED BICYCLIC HETEROCYCLIC DERIVATIVES AS PEST CONTROL AGENTS BAYER AKTIENGESELLSCHAFT (DE) 2019-08-29 WO disclosed
EP-3523299-A1 2-(HET)ARYL-SUBSTITUTED CONDENSED BICYCLIC HETEROCYCLE DERIVATIVES AS PEST CONTROL AGENTS Bayer CropScience Aktiengesellschaft (DE) 2019-08-14 EP disclosed
EP-3515921-A1 PYRAZOLO [1,5-A]PYRIDINE DERIVATIVES AND THEIR USE AS PESTICIDES Bayer CropScience Aktiengesellschaft (DE) 2019-07-31 EP disclosed
EP-3319943-B1 NITROGEN-CONTAINING HETEROCYCLES AS PESTICIDES BAYER CROPSCIENCE AG (DE) 2019-06-26 EP disclosed
EP-3497102-A1 CONDENSED BICYCLIC HETEROCYCLE DERIVATIVES AS PEST CONTROL AGENTS Bayer CropScience Aktiengesellschaft (DE) 2019-06-19 EP disclosed
EP-3487860-A1 CONDENSED BICYCLIC HETEROCYCLE DERIVATIVES AS PEST CONTROL AGENTS Bayer CropScience Aktiengesellschaft (DE) 2019-05-29 EP disclosed
EP-3484877-A1 BICYCLIC COMPOUNDS AS PEST CONTROL AGENTS Bayer CropScience Aktiengesellschaft (DE) 2019-05-22 EP disclosed
EP-3419418-A1 SOLVENT-FREE FORMULATIONS OF LOW-MELTING ACTIVE SUBSTANCES Bayer CropScience Aktiengesellschaft (DE) 2019-01-02 EP disclosed
EP-3402797-A1 HETEROCYCLENE DERIVATIVES AS PEST CONTROL AGENTS Bayer CropScience AG (DE) 2018-11-21 EP disclosed
EP-3356362-A1 2-(HET)ARYL-SUBSTITUTED CONDENSED BICYCLIC HETEROCYCLIC DERIVATIVES AS PEST CONTROL AGENTS Bayer CropScience Aktiengesellschaft (DE) 2018-08-08 EP disclosed