SCHEMBL2045341

SCHEMBL2045341

CCn1nnc(CCl)n1.CCn1nnc(CCl)n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.40
LMNA P02545 1/20 0.40
HSD17B10 Q99714 2/20 0.36
PKM P14618 2/20 0.36
ATM Q13315 1/20 0.36
CHRM2 P08172 2/20 0.34
CHRM3 P20309 1/20 0.34
L3MBTL1 Q9Y468 2/20 0.34
ESR1 P03372 1/20 0.34
POLB P06746 1/20 0.34
ESR2 Q92731 1/20 0.34
HTR1A P08908 1/20 0.33
HTR2C P28335 1/20 0.33
TRPM8 Q7Z2W7 2/20 0.32
NPC1 O15118 2/20 0.32
RAB9A P51151 2/20 0.32
ALDH1A1 P00352 2/20 0.31
TP53 P04637 1/20 0.31
MAPK1 P28482 1/20 0.31
HTT P42858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2049146 1.00
SCHEMBL4412024 0.81
SCHEMBL23277296 0.79
SCHEMBL4409234 0.77 SMN1; SMN2 (0.40) SMN1; SMN2LMNAHSD17B10PKMATM
SCHEMBL1302329 0.77
SCHEMBL4409055 0.74 SMN1; SMN2 (0.42) SMN1; SMN2LMNAHSD17B10PKMATM
SCHEMBL1302376 0.74 SMN1; SMN2 (0.46) SMN1; SMN2LMNAHSD17B10PKMATM
SCHEMBL4408760 0.74 LMNA (0.38) SMN1; SMN2LMNAHSD17B10PKMATM
SCHEMBL4407234 0.74 TRPV1 (0.38) SMN1; SMN2LMNAHSD17B10PKMATM
SCHEMBL4411011 0.72 GPR84 (0.38) SMN1; SMN2LMNAHSD17B10PKMATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2513119-A1 3,4,4A,10B-TETRAHYDRO-1H-THIOPYRANO-[4, 3-c]ISOQUINOLINE DERIVATIVES Nycomed GmbH (DE) 2012-10-24 EP disclosed
WO-2011073231-A1 3,4,4A,10B-TETRAHYDRO-1H-THIOPYRANO-[4, 3-c] ISOQUINOLINE DERIVATIVES NYCOMED GMBH (DE) 2011-06-23 WO disclosed