SCHEMBL2045458

SCHEMBL2045458

O=[N+]([O-])c1c(O)cccc1C1CCOO1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GPR35 Q9HC97 2/20 0.45
S100A4 P26447 2/20 0.35
STS P08842 2/20 0.33
HSP90AA1 P07900 2/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
TLR9 Q9NR96 1/20 0.33
MCL1 Q07820 1/20 0.33
ALDH1A1 P00352 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
GAA P10253 3/20 0.32
ESR1 P03372 1/20 0.31
ESR2 Q92731 1/20 0.31
MAPT P10636 1/20 0.31
CSNK2A2 P19784 1/20 0.31
CSNK2B P67870 1/20 0.31
CSNK2A1 P68400 1/20 0.31
CSNK2A3 Q8NEV1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6521534 0.81 GPR35 (0.46) GPR35S100A4STSHSP90AA1MEN1
SCHEMBL6184572 0.77 TRPA1 (0.38) MEN1KMT2AESR1ESR2MAPT
SCHEMBL19899567 0.77 GPR35 (0.55) GPR35S100A4STSHSP90AA1MEN1
SCHEMBL6184401 0.76 AR (0.41) MEN1KMT2AALDH1A1TDP1GAA
SCHEMBL8935115 0.76 DNMT3B (0.40) MEN1KMT2AALDH1A1TDP1GAA
SCHEMBL6184452 0.74 ESR1 (0.32) MEN1KMT2AESR1ESR2
SCHEMBL6186797 0.71 CA1 (0.38) ALDH1A1ESR1ESR2MAPT
SCHEMBL31473755 0.70 GPR35 (0.44) GPR35S100A4STSMEN1KMT2A
SCHEMBL70533 0.70 GPR35 (0.75) GPR35S100A4ALDH1A1TDP1ESR1
SCHEMBL28687501 0.69 GPR35 (0.42) GPR35S100A4HSP90AA1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011140202-A2 MIF MODULATORS YALE UNIVERSITY (US) 2011-11-10 WO disclosed
EP-2326631-A2 MIF MODULATORS Yale University (US) 2011-06-01 EP disclosed
WO-2010021693-A2 MIF MODULATORS YALE UNIVERSITY (US) 2010-02-25 WO disclosed
EP-1581218-A1 EPOTHILONE ANALOGS FOR SITE SPECIFIC DELIVERY IN THE TREATMENT OF PROLIFERATIVE DISEASES Schering AG (DE) 2005-10-05 EP disclosed
WO-2004050089-A1 EPOTHILONE ANALOGS FOR SITE SPECIFIC DELIVERY IN THE TREATMENT OF PROLIFERATIVE DISEASES SCHERING AG (DE) 2004-06-17 WO disclosed