SCHEMBL20456403

SCHEMBL20456403

CS(=O)(=O)c1nc2cccc(N)c2c(=O)n1C1CCC(=O)NC1=O

nearest known ligand 0.74

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 20/20 0.74
DDB1 Q16531 19/20 0.74
IKZF3 Q9UKT9 6/20 0.74
TNF P01375 3/20 0.74
IL1B P01584 3/20 0.74
IKZF1 Q13422 2/20 0.47
TBXA2R P21731 1/20 0.47
BRD4 O60885 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Avadomide SCHEMBL15120730 0.85 CRBN (1.00) CRBNDDB1IKZF3TNFIL1B
Avadomide SCHEMBL29442249 0.85 CRBN (1.00) CRBNDDB1IKZF3TNFIL1B
Avadomide SCHEMBL29359950 0.85 CRBN (1.00) CRBNDDB1IKZF3TNFIL1B
Avadomide SCHEMBL634577 0.85 CRBN (1.00) CRBNDDB1IKZF3TNFIL1B
Avadomide SCHEMBL282749 0.85 CRBN (1.00) CRBNDDB1IKZF3TNFIL1B
SCHEMBL20456410 0.84 CRBN (0.52) CRBNDDB1IKZF3TNFIL1B
Avadomide SCHEMBL12099722 0.84 CRBN (0.98) CRBNDDB1IKZF3TNFIL1B
Avadomide SCHEMBL29519996 0.84 CRBN (0.98) CRBNDDB1IKZF3TNFIL1B
Avadomide SCHEMBL29520051 0.84 CRBN (0.98) CRBNDDB1IKZF3TNFIL1B
Avadomide SCHEMBL15515920 0.84 CRBN (0.98) CRBNDDB1IKZF3TNFIL1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018144445-A1 METHODS FOR TREATING HEMATOLOGICAL CANCER AND THE USE OF BIOMARKERS AS A PREDICTOR FOR RESPONSIVENESS TO TREATMENT COMPOUNDS CELGENE CORPORATION (US) 2018-08-09 WO disclosed