SCHEMBL20459986

SCHEMBL20459986

Clc1ncc(Br)nc1N1CCCCC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.42
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
GFER P55789 2/20 0.41
ALDH1A1 P00352 4/20 0.40
MAPK1 P28482 2/20 0.40
MAPT P10636 3/20 0.39
GAA P10253 1/20 0.39
LMNA P02545 3/20 0.38
SLC9A5 Q14940 2/20 0.38
PLAU P00749 2/20 0.38
ADORA2A P29274 2/20 0.38
TDP1 Q9NUW8 2/20 0.38
NPC1 O15118 1/20 0.38
TP53 P04637 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
SLC9A1 P19634 1/20 0.38
ADORA2B P29275 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14725974 0.83 ALDH1A1 (0.48) TSHRALDH1A1MAPK1MAPTGAA
SCHEMBL2317513 0.80 CYP1A2 (0.47) TSHRALDH1A1MAPK1MAPTADORA2A
SCHEMBL2321134 0.78 TSHR (0.44) TSHRGFERALDH1A1MAPK1MAPT
SCHEMBL22234855 0.78 MAPT (0.49) TSHRGFERALDH1A1MAPK1MAPT
SCHEMBL2322572 0.78 TSHR (0.44) TSHRGFERALDH1A1MAPK1MAPT
SCHEMBL2324009 0.76 ALDH1A1 (0.42) TSHRGFERALDH1A1MAPK1MAPT
SCHEMBL3815039 0.73 MAPT (0.46) TSHRMEN1KMT2AALDH1A1MAPK1
SCHEMBL2321291 0.72 ROCK2 (0.60)
SCHEMBL2320168 0.72 ROCK2 (0.60)
SCHEMBL19240314 0.71 GFER (0.47) TSHRMEN1KMT2AGFERALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2867232-B1 5-AZAINDAZOLE COMPOUNDS AND METHODS OF USE HOFFMANN LA ROCHE (CH) 2018-08-08 EP disclosed