SCHEMBL20460745

SCHEMBL20460745

Cc1nc2c(n1C)CCN(C(=O)C(C)C)C2

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 12/20 0.44
KCNH2 Q12809 2/20 0.42
P2RX7 Q99572 2/20 0.39
DPP4 P27487 2/20 0.38
DPP8 Q6V1X1 2/20 0.38
DPP7 Q9UHL4 2/20 0.38
DPP9 Q86TI2 1/20 0.38
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35
CNR2 P34972 1/20 0.33
GPR6 P46095 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23374970 0.83 CCR5 (0.42) CCR5KCNH2P2RX7DPP4DPP8
SCHEMBL23374968 0.82 P2RX7 (0.37) CCR5KCNH2P2RX7DPP4DPP8
SCHEMBL8277482 0.72 PDCD1 (0.38) P2RX7
SCHEMBL16219043 0.71 DPP4 (0.49) DPP4DPP8DPP7DPP9
SCHEMBL16219073 0.71 GRM5 (0.42) CCR5DPP4DPP8DPP7DPP9
SCHEMBL16219076 0.71 JAK2 (0.41) KCNH2DPP4DPP8GPR6
SCHEMBL23374967 0.71 DPP4 (0.30) DPP4DPP8DPP7DPP9
SCHEMBL23374979 0.71 PDCD1 (0.48) DPP4DPP8DPP7DPP9CNR2
SCHEMBL16219049 0.71 CREBBP (0.42)
SCHEMBL21620980 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3091013-B1 1-(3-AMINOPROPYL) SUBSTITUTED CYCLIC AMINE COMPOUNDS, PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL COMPOSITIONS AND USES THEREOF SHANGHAI INST MATERIA MEDICA CAS (CN) 2018-08-08 EP disclosed