SCHEMBL20478682

SCHEMBL20478682

NC(=O)C1(S(=O)(=O)Cc2ccccc2)CCc2ccccc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 4/20 0.38
ALDH1A1 P00352 3/20 0.38
TSHR P16473 2/20 0.38
HDAC9 Q9UKV0 1/20 0.38
TP53 P04637 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
F2 P00734 1/20 0.38
PRSS1 P07477 1/20 0.38
PRSS2 P07478 1/20 0.38
PRSS3 P35030 1/20 0.38
GLA P06280 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA5A P35218 1/20 0.37
CA9 Q16790 1/20 0.37
HCAR2 Q8TDS4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2172389 0.80 HDAC9 (0.40) TSHRHDAC9HCAR2OPRL1
SCHEMBL22572200 0.73 ITGB1 (0.48) ALDH1A1TSHRF2PRSS1PRSS2
SCHEMBL315669 0.72 GAA (0.42) HDAC9
SCHEMBL315173 0.72 GAA (0.42) HDAC9
SCHEMBL20478817 0.70 F2 (0.42) TSHRF2PRSS1PRSS2PRSS3
SCHEMBL28136981 0.68 KDM1A (0.47) TSHRHDAC9HCAR2OPRL1
SCHEMBL17335394 0.68 KDM1A (0.46) TSHRHDAC9HCAR2OPRL1
SCHEMBL7398453 0.67 SIGMAR1 (0.44) SIGMAR1TSHRHDAC9TP53CYP1A2
SCHEMBL29677121 0.66 KDM4E (0.45) ALDH1A1TSHRHDAC9CYP1A2CYP2C19
SCHEMBL5147955 0.66 KDM1A (0.44) TSHRHDAC9HCAR2OPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180244611-A1 Modulators of the Cystic Fibrosis Transmembrane Conductance Regulator Protein and Methods of Use ABBVIE S.Á.R.L. (LU) 2018-08-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180244611-A1 Modulators of the Cystic Fibrosis Transmembrane Conductance Regulator Protein and Methods of Use CFTR, CLCN2, SCNN1G SIGMAR1 2473/4885ALDH1A1 4131/4885TSHR 2071/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.