SCHEMBL20488709

SCHEMBL20488709

[CH2]C#Cc1cccc(Cl)c1

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.53
GRM5 P41594 9/20 0.49
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.40
PTGDR2 Q9Y5Y4 1/20 0.40
ALDH1A1 P00352 1/20 0.39
TSHR P16473 1/20 0.39
MAOB P27338 1/20 0.39
PNMT P11086 1/20 0.35
HAO1 Q9UJM8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4562631 0.85 KCNH2 (0.67) KCNH2GRM5CYP2D6CYP2C9PTGDR2
SCHEMBL30707869 0.85 KCNH2 (0.67) KCNH2GRM5CYP2D6CYP2C9PTGDR2
Charcoal, Activated SCHEMBL31286308 0.83 KCNH2 (0.64) KCNH2GRM5CYP2D6CYP2C9PTGDR2
SCHEMBL25490062 0.79 KCNH2 (0.55) KCNH2GRM5CYP2D6CYP2C9PTGDR2
SCHEMBL29978649 0.79 KCNH2 (0.55) KCNH2GRM5CYP2D6CYP2C9PTGDR2
SCHEMBL718734 0.79 KCNH2 (0.55) KCNH2GRM5CYP2D6CYP2C9PTGDR2
SCHEMBL717449 0.79 KCNH2 (0.60) KCNH2GRM5CYP2D6CYP2C9PTGDR2
SCHEMBL21252707 0.77 KCNH2 (0.53) KCNH2GRM5CYP2D6CYP2C9PTGDR2
SCHEMBL2697031 0.77 KCNH2 (0.58) KCNH2GRM5CYP2D6CYP2C9PTGDR2
SCHEMBL30081497 0.77 KCNH2 (0.58) KCNH2GRM5CYP2D6CYP2C9PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018157800-A1 MLKL INHIBITORS NATIONAL INSTITUTE OF BIOLOGICAL SCIENCES, BEIJING (CN) 2018-09-07 WO disclosed