SCHEMBL20495178

SCHEMBL20495178

O=CC[C@H](Br)c1ccc(F)cc1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.34
TDO2 P48775 2/20 0.34
HDAC3 O15379 1/20 0.34
HDAC4 P56524 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC7 Q8WUI4 1/20 0.34
HDAC2 Q92769 1/20 0.34
HDAC10 Q969S8 1/20 0.34
HDAC11 Q96DB2 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
HDAC9 Q9UKV0 1/20 0.34
HDAC5 Q9UQL6 1/20 0.34
AOC3 Q16853 2/20 0.33
SLC6A3 Q01959 1/20 0.33
GABBR2 O75899 1/20 0.33
GABBR1 Q9UBS5 1/20 0.33
PTPN1 P18031 1/20 0.32
HTT P42858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1150763 1.00 IDO1 (0.34) IDO1TDO2HDAC3HDAC4HDAC1
SCHEMBL26106019 0.80 IDO1 (0.32) IDO1TDO2HDAC3HDAC4HDAC1
SCHEMBL17763415 0.78 CES2 (0.41)
SCHEMBL65457 0.78 CACNA2D1 (0.37) IDO1TDO2HDAC3HDAC4HDAC1
SCHEMBL3136328 0.78 GABBR2 (0.43) IDO1TDO2HDAC3HDAC4HDAC1
SCHEMBL12860041 0.77 HIF1A (0.31) IDO1TDO2HDAC3HDAC4HDAC1
SCHEMBL27629443 0.77 IDO1 (0.35) IDO1TDO2HDAC3HDAC4HDAC1
SCHEMBL15577528 0.76 HTR2A (0.41) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL6221926 0.75 IDO1 (0.34) IDO1TDO2HDAC3HDAC4HDAC1
SCHEMBL31378985 0.75 AOC3 (0.47) IDO1HDAC3HDAC4HDAC1HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018165520-A1 METALLOENZYME INHIBITOR COMPOUNDS VPS-3, INC. (US) 2018-09-13 WO disclosed