SCHEMBL20503249

SCHEMBL20503249

Cc1nn(-c2ccc(CC(C)C)cc2)cc1C(=O)O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALKBH1 Q13686 1/20 0.45
PTGS2 P35354 4/20 0.42
PTGS1 P23219 3/20 0.42
LMNA P02545 3/20 0.42
CYP2C9 P11712 2/20 0.42
AKR1C3 P42330 2/20 0.42
CXCR1 P25024 2/20 0.42
CXCR2 P25025 2/20 0.42
AKR1C2 P52895 2/20 0.42
ALB P02768 1/20 0.42
ESR1 P03372 1/20 0.42
ALOX5 P09917 1/20 0.42
RARB P10826 1/20 0.42
ADRB3 P13945 1/20 0.42
NFKB1 P19838 1/20 0.42
HTR2A P28223 1/20 0.42
NR1I3 Q14994 1/20 0.42
SLC22A6 Q4U2R8 1/20 0.42
CXCL8 P10145 1/20 0.42
TSHR P16473 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20556573 0.85 MAPT (0.46) PTGS2CXCR1CXCR2ENPP3ALPL
SCHEMBL4298023 0.79 ALDH1A1 (0.59) ALKBH1LMNAALDH1A1MAPTKDM4E
SCHEMBL6052147 0.78 MEN1 (0.53) ALKBH1LMNAALDH1A1MAPTKDM4E
SCHEMBL6052366 0.78 NOTUM (0.49) LMNAALDH1A1MAPTKDM4EMEN1
SCHEMBL6052337 0.78 NOTUM (0.49) ALKBH1LMNAALDH1A1MAPTKDM4E
SCHEMBL6052367 0.75 L3MBTL1 (0.63) ALKBH1LMNAALDH1A1MAPTKDM4E
SCHEMBL29333627 0.74 ALDH1A1 (0.42) ALKBH1LMNAALDH1A1MAPTKDM4E
SCHEMBL15167860 0.74 CA12 (0.63) PTGS2PTGS1LMNAALDH1A1MAPT
SCHEMBL20552556 0.71 ALDH1A1 (0.44) ALKBH1LMNAALDH1A1MAPTKDM4E
SCHEMBL10321717 0.71 ALDH1A1 (0.54) LMNATSHRALDH1A1MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3377473-A1 MACROCYCLIC BROAD SPECTRUM ANTIBIOTICS RQX Pharmaceuticals, Inc. (US) 2018-09-26 EP disclosed