Dimethyl Maleate

Dimethyl Maleate

SCHEMBL20508358

CCCC.COC(=O)/C=C\C(=O)OC

nearest known ligand 0.77

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

KEAP1

The experimentally established mechanism targets of Dimethyl Maleate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 known ✓ Q14145 1/20 0.77
HCAR2 Q8TDS4 7/20 0.77
NFE2L2 Q16236 2/20 0.77
ATM Q13315 1/20 0.48
GFPT1 Q06210 1/20 0.44
MAPT P10636 2/20 0.42
ALDH1A1 P00352 2/20 0.42
KDM4E B2RXH2 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
TYR P14679 1/20 0.40
CA7 P43166 1/20 0.40
CA9 Q16790 1/20 0.40
CA14 Q9ULX7 1/20 0.40
RAB9A P51151 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
ALOX15 P16050 1/20 0.39
RECQL P46063 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Monomethyl Fumarate SCHEMBL11129720 0.90 HCAR2 (0.81) HCAR2NFE2L2KEAP1ATMGFPT1
Dimethyl Maleate SCHEMBL6417885 0.88 HCAR2 (0.77) HCAR2NFE2L2KEAP1ATMGFPT1
Dimethyl Fumarate SCHEMBL41835 0.87 NFE2L2 (1.00) HCAR2NFE2L2KEAP1GFPT1MAPT
Dimethyl Maleate SCHEMBL75864 0.87 NFE2L2 (1.00) HCAR2NFE2L2KEAP1GFPT1MAPT
Dimethyl Fumarate SCHEMBL41836 0.87 NFE2L2 (1.00) HCAR2NFE2L2KEAP1GFPT1MAPT
Dimethyl Fumarate SCHEMBL28128958 0.87 NFE2L2 (1.00) HCAR2NFE2L2KEAP1GFPT1MAPT
Dimethyl Fumarate SCHEMBL11668350 0.87 NFE2L2 (1.00) HCAR2NFE2L2KEAP1GFPT1MAPT
Dimethyl Maleate SCHEMBL27720952 0.87 NFE2L2 (1.00) HCAR2NFE2L2KEAP1GFPT1MAPT
SCHEMBL14282529 0.85 NFE2L2 (0.81) HCAR2NFE2L2KEAP1GFPT1MAPT
SCHEMBL16257486 0.85 NFE2L2 (0.81) HCAR2NFE2L2KEAP1GFPT1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180277881-A1 SECONDARY BATTERY, BATTERY PACK, ELECTRIC VEHICLE, POWER STORAGE SYSTEM, ELECTRIC TOOL, ELECTRONIC DEVICE MURATA MANUFACTURING CO., LTD. (JP) 2018-09-27 US disclosed