SCHEMBL20510885

SCHEMBL20510885

C=CCN[C@@H](CO)c1ccc(Br)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 2/20 0.40
SMN1; SMN2 Q16637 3/20 0.37
LMNA P02545 4/20 0.36
TGM2 P21980 2/20 0.36
F13A1 P00488 1/20 0.36
TGM1 P22735 1/20 0.36
TGM3 Q08188 1/20 0.36
ATM Q13315 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
HTT P42858 3/20 0.34
NPC1 O15118 1/20 0.34
STAT1 P42224 1/20 0.34
RAB9A P51151 1/20 0.34
CNR1 P21554 2/20 0.33
CYP1A2 P05177 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
S1PR3 Q99500 1/20 0.33
MMP9 P14780 2/20 0.32
KDM4E B2RXH2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3567880 0.86 SMN1; SMN2 (0.49) CYP2C19SMN1; SMN2LMNATGM2F13A1
SCHEMBL6389932 0.82 SMN1; SMN2 (0.49) CYP2C19SMN1; SMN2ATML3MBTL1KDM4E
SCHEMBL1978925 0.72 CYP1A2 (0.42) CYP2C19SMN1; SMN2CNR1CYP1A2ALDH1A1
SCHEMBL323957 0.71 ADRB2 (0.56) SMN1; SMN2ATML3MBTL1HTTCNR1
SCHEMBL24325919 0.69 SMN1; SMN2 (0.69) CYP2C19SMN1; SMN2ATML3MBTL1RAB9A
SCHEMBL2290184 0.69 KDM4E (0.44) CYP2C19SMN1; SMN2LMNATGM2F13A1
SCHEMBL2291816 0.69 KDM4E (0.44) CYP2C19SMN1; SMN2LMNATGM2F13A1
SCHEMBL1554805 0.68 CYP1A2 (0.47) CYP2C19SMN1; SMN2CNR1CYP1A2MEN1
SCHEMBL17710307 0.68 CYP1A2 (0.47) CYP2C19SMN1; SMN2CNR1CYP1A2MEN1
Hydrochloric Acid SCHEMBL18553838 0.68 SMN1; SMN2 (0.45) CYP2C19SMN1; SMN2LMNAATML3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3600286-A1 COMPOUNDS AND METHODS FOR THE TREATMENT OF PARASITIC DISEASES The Broad Institute, Inc. (US) 2020-02-05 EP disclosed
WO-2018175385-A1 COMPOUNDS AND METHODS FOR THE TREATMENT OF PARASITIC DISEASES THE BROAD INSTITUTE, INC. (US) 2018-09-27 WO disclosed