SCHEMBL20512401

SCHEMBL20512401

O=C1CCC(CCOC(c2ccccc2)(c2ccccc2)c2ccccc2)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 1/20 0.47
SLC6A1 P30531 3/20 0.42
CYP2C9 P11712 2/20 0.42
TSHR P16473 2/20 0.42
CYP2C19 P33261 2/20 0.42
ALOX15 P16050 1/20 0.42
DUT P33316 1/20 0.40
TK2 O00142 6/20 0.37
TK1 P04183 2/20 0.36
SLC6A11 P48066 1/20 0.36
HRH4 Q9H3N8 1/20 0.35
CHRM2 P08172 2/20 0.33
CHRM4 P08173 2/20 0.33
CHRM1 P11229 2/20 0.33
CHRM3 P20309 2/20 0.33
SLC22A1 O15245 1/20 0.33
MLNR O43193 1/20 0.33
NR1I2 O75469 1/20 0.33
TP53 P04637 1/20 0.33
ADRB2 P07550 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL99301 0.79 KIF11 (0.49) KIF11SLC6A1CYP2C9TSHRCYP2C19
SCHEMBL99300 0.79 KIF11 (0.49) KIF11SLC6A1CYP2C9TSHRCYP2C19
SCHEMBL20512399 0.78 KIF11 (0.45) KIF11SLC6A1CYP2C9TSHRCYP2C19
SCHEMBL1197663 0.77 TSHR (0.44) CYP2C9TSHRCYP2C19CYP3A4DRD2
SCHEMBL5519659 0.77 TEAD1 (0.52)
SCHEMBL99951 0.74 KIF11 (0.41) KIF11SLC6A1CYP2C9TSHRCYP2C19
SCHEMBL99952 0.74 KIF11 (0.41) KIF11SLC6A1CYP2C9TSHRCYP2C19
SCHEMBL11275984 0.72 KIF11 (0.74) KIF11SLC6A1CYP2C9TSHRCYP2C19
SCHEMBL25738193 0.72 ALDH1A1 (0.30) KMT2A
SCHEMBL9481131 0.71 KIF11 (0.52) KIF11SLC6A1CYP2C9TSHRCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3184526-B1 PYRROLO[2,3-D]PYRIMIDINE DERIVATIVES AS JANUS KINASE INHIBITOR INCYTE HOLDINGS CORP (US) 2018-10-03 EP disclosed