SCHEMBL20523609

SCHEMBL20523609

CCCS(=O)(=O)Nc1ccc(-c2cc(-c3ccc(N4CCN(C(=O)O)CC4)cc3)cnc2Cl)cc1OC

nearest known ligand 0.65

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NOD2 Q9HC29 14/20 0.65
RIPK2 O43353 14/20 0.56
ACVR1 Q04771 12/20 0.56
NOD1 Q9Y239 1/20 0.48
TGFBR1 P36897 2/20 0.47
FYN P06241 1/20 0.43
MAP4K1 Q92918 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21630350 0.90 NOD2 (0.61) NOD2RIPK2ACVR1NOD1TGFBR1
SCHEMBL21630369 0.86 NOD2 (0.68) NOD2RIPK2ACVR1NOD1TGFBR1
SCHEMBL21630433 0.86 NOD2 (0.65) NOD2RIPK2ACVR1NOD1TGFBR1
SCHEMBL21630382 0.80 NOD2 (0.63) NOD2RIPK2ACVR1TGFBR1
SCHEMBL20523635 0.79 NOD2 (1.00) NOD2RIPK2ACVR1NOD1TGFBR1
SCHEMBL21630356 0.76 LMNA (0.51) NOD2RIPK2ACVR1
SCHEMBL20523500 0.76 ACVR1 (0.62) NOD2RIPK2ACVR1TGFBR1FYN
SCHEMBL21630387 0.76 ACVR1 (0.51) NOD2RIPK2ACVR1TGFBR1FYN
SCHEMBL21630442 0.76 NOD2 (0.54) NOD2RIPK2ACVR1TGFBR1FYN
SCHEMBL20523650 0.74 KMT2A (0.47) ACVR1TGFBR1FYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3600307-A1 COMPOSITIONS FOR USE IN METHODS OF INHIBITING PROTEIN KINASES University of Houston System (US) 2020-02-05 EP disclosed
WO-2018183633-A1 COMPOSITIONS FOR USE IN METHODS OF INHIBITING PROTEIN KINASES UNIVERSITY OF HOUSTON SYSTEM (US) 2018-10-04 WO disclosed