SCHEMBL20524183

SCHEMBL20524183

CC(C)(C)[Si](Oc1ccc(C2CCC(=CC(=O)O)CC2)cc1)(c1ccccc1)c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 2/20 0.40
MAPK1 P28482 1/20 0.35
MAPK14 Q16539 1/20 0.35
HCAR2 Q8TDS4 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
CASP1 P29466 2/20 0.31
CCR1 P32246 2/20 0.31
HSD11B1 P28845 1/20 0.31
MRGPRX4 Q96LA9 1/20 0.31
LMNA P02545 2/20 0.30
CYP2C9 P11712 1/20 0.30
TSHR P16473 1/20 0.30
BLM P54132 1/20 0.30
PPARA Q07869 1/20 0.30
KDM4E B2RXH2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18258349 0.87 ESR2 (0.59) ESR2MAPK1MAPK14RAB9ALMNA
SCHEMBL18244774 0.84 ESR2 (0.50) ESR2MAPK1MAPK14
SCHEMBL18244723 0.83 ESR2 (0.42) ESR2MAPK1MAPK14
SCHEMBL12919164 0.70 CA1 (0.46) TSHR
SCHEMBL16743002 0.70 ESR2 (0.59) ESR2RAB9ALMNAKDM4E
SCHEMBL2257887 0.70 ESR2 (0.62) ESR2CYP2C9
SCHEMBL17070013 0.69 ELANE (0.54) PPARA
SCHEMBL863103 0.69 MAOB (0.46) NPC1RAB9ALMNACYP2C9PPARA
SCHEMBL704145 0.69 CA4 (0.37) ESR2MAPK1TSHR
SCHEMBL7096596 0.68 ESR2 (0.46) ESR2LMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3601204-A1 SUBSTITUTED (4'-HYDROXYPHENYL)CYCLOALKANE AND (4'-HYDROXYPHENYL)CYCLOALKENE COMPOUNDS AND USES THEREOF AS SELECTIVE AGONISTS OF THE ESTROGEN RECEPTOR BETA ISOFORM FOR ENHANCED MEMORY CONSOLIDATION Marquette University (US) 2020-02-05 EP disclosed
WO-2018183800-A1 SUBSTITUTED (4'-HYDROXYPHENYL)CYCLOALKANE AND (4'-HYDROXYPHENYL)CYCLOALKENE COMPOUNDS AND USES THEREOF AS SELECTIVE AGONISTS OF THE ESTROGEN RECEPTOR BETA ISOFORM FOR ENHANCED MEMORY CONSOLIDATION MARQUETTE UNIVERSITY (US) 2018-10-04 WO disclosed