SCHEMBL2052497

SCHEMBL2052497

O=C(On1cnc2c(NCCc3cc(F)c4ccnnc4c3-c3cc(F)cc(F)c3)ncnc21)C(F)(F)F

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TMIGD3 P0DMS9 2/20 0.33
ADORA2A P29274 2/20 0.33
ADORA1 P30542 2/20 0.33
ADORA2B P29275 1/20 0.33
PDE4A P27815 1/20 0.31
PDE4B Q07343 1/20 0.31
PDE4C Q08493 1/20 0.31
PDE4D Q08499 1/20 0.31
ALDH1A1 P00352 1/20 0.30
POLB P06746 1/20 0.30
PKM P14618 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2051000 0.86 PIK3CD (0.33) TMIGD3ADORA2AADORA1ADORA2B
SCHEMBL2164179 0.82 PIK3CD (0.41)
SCHEMBL2038100 0.79 PIK3CD (0.41) ADORA2AADORA1ADORA2B
Trifluoroacetic Acid SCHEMBL2052496 0.79 PIK3CD (0.35)
SCHEMBL2165865 0.70 PIK3CD (0.47)
SCHEMBL9960866 0.70 LMNA (0.36) ALDH1A1
SCHEMBL2016719 0.68 PIK3CD (0.47)
SCHEMBL2017997 0.67 PIK3CD (0.39)
SCHEMBL2012486 0.67 PIK3CD (0.46)
Trifluoroacetic Acid SCHEMBL2050998 0.65 PIK3CD (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011075630-A1 SUBSTITUTED FUSED ARYL AND HETEROARYL DERIVATIVES AS PI3K INHIBITORS INCYTE CORPORATION (US) 2011-06-23 WO disclosed